Search details
1.
ChemFH: an integrated tool for screening frequent false positives in chemical biology and drug discovery.
Nucleic Acids Res
; 2024 May 23.
Article
in English
| MEDLINE | ID: mdl-38783035
2.
ADMETlab 3.0: an updated comprehensive online ADMET prediction platform enhanced with broader coverage, improved performance, API functionalityĀ and decision support.
Nucleic Acids Res
; 2024 Apr 04.
Article
in English
| MEDLINE | ID: mdl-38572755
3.
Enhancing Multi-species Liver Microsomal Stability Prediction through Artificial Intelligence.
J Chem Inf Model
; 64(8): 3222-3236, 2024 Apr 22.
Article
in English
| MEDLINE | ID: mdl-38498003
4.
Evaluation of Platensimycin and Platensimycin-Inspired Thioether Analogues against Methicillin-Resistant Staphylococcus aureus in Topical and Systemic Infection Mouse Models.
Mol Pharm
; 16(7): 3065-3071, 2019 07 01.
Article
in English
| MEDLINE | ID: mdl-31244223
5.
Stereoselective functionalization of platensimycin and platencin by sulfa-Michael/aldol reactions.
Org Biomol Chem
; 17(17): 4261-4272, 2019 04 24.
Article
in English
| MEDLINE | ID: mdl-30816397
6.
Design, synthesis and biological Evaluation of Dual acetyl cholinesterase and beta-secretase inhibitors in treatment for alzheimer's Disease.
Pak J Pharm Sci
; 32(5): 2091-2098, 2019 Sep.
Article
in English
| MEDLINE | ID: mdl-31813875
7.
Biomimetic Stereoselective Sulfa-Michael Addition Leads to Platensimycin and Platencin Sulfur Analogues against Methicillin-Resistant Staphylococcus aureus.
J Nat Prod
; 81(2): 316-322, 2018 02 23.
Article
in English
| MEDLINE | ID: mdl-29389125
8.
Butyrylcholinesterase K variant and Alzheimer's disease risk: a meta-analysis.
Med Sci Monit
; 21: 1408-13, 2015 May 16.
Article
in English
| MEDLINE | ID: mdl-25978873
9.
Enhancing Molecular Property Prediction through Task-Oriented Transfer Learning: Integrating Universal Structural Insights and Domain-Specific Knowledge.
J Med Chem
; 2024 May 15.
Article
in English
| MEDLINE | ID: mdl-38748846
10.
Structure-Activity Relationship Studies of Venglustat on NTMT1 Inhibition.
J Med Chem
; 66(2): 1601-1615, 2023 01 26.
Article
in English
| MEDLINE | ID: mdl-36634151
11.
A unique binding pocket induced by a noncanonical SAH mimic to develop potent and selective PRMT inhibitors.
Acta Pharm Sin B
; 13(12): 4893-4905, 2023 Dec.
Article
in English
| MEDLINE | ID: mdl-38045046
12.
Comparative Study of Adenosine Analogs as Inhibitors of Protein Arginine Methyltransferases and a Clostridioides difficile-Specific DNA Adenine Methyltransferase.
ACS Chem Biol
; 18(4): 734-745, 2023 04 21.
Article
in English
| MEDLINE | ID: mdl-37082867
13.
Morphing Natural Product Platensimycin via Heck, Sonogashira, and One-Pot Sonogashira/Cycloaddition Reactions to Produce Antibiotics with In Vivo Activity.
Antibiotics (Basel)
; 11(4)2022 Mar 23.
Article
in English
| MEDLINE | ID: mdl-35453177
14.
Venglustat Inhibits Protein N-Terminal Methyltransferase 1 in a Substrate-Competitive Manner.
J Med Chem
; 65(18): 12334-12345, 2022 09 22.
Article
in English
| MEDLINE | ID: mdl-36074125
15.
Structure-based Discovery of Cell-Potent Peptidomimetic Inhibitors for Protein N-Terminal Methyltransferase 1.
ACS Med Chem Lett
; 12(3): 485-493, 2021 Mar 11.
Article
in English
| MEDLINE | ID: mdl-33738076
16.
Discovery of a potent and dual-selective bisubstrate inhibitor for protein arginine methyltransferase 4/5.
Acta Pharm Sin B
; 11(9): 2709-2718, 2021 Sep.
Article
in English
| MEDLINE | ID: mdl-34589391
17.
Novel Bisubstrate Inhibitors for Protein N-Terminal Acetyltransferase D.
J Med Chem
; 64(12): 8263-8271, 2021 06 24.
Article
in English
| MEDLINE | ID: mdl-34110812
18.
Semisynthesis and Biological Evaluation of Platencin Thioether Derivatives: Dual FabF and FabH Inhibitors against MRSA.
ACS Med Chem Lett
; 12(3): 433-442, 2021 Mar 11.
Article
in English
| MEDLINE | ID: mdl-33738071
19.
Late-Stage Functionalization of Platensimycin Leading to Multiple Analogues with Improved Antibacterial Activity in Vitro and in Vivo.
J Med Chem
; 62(14): 6682-6693, 2019 07 25.
Article
in English
| MEDLINE | ID: mdl-31265289
20.
Semisynthesis and Biological Evaluation of Platensimycin Analogues with Varying Aminobenzoic Acids.
ChemistrySelect
; 3(44): 12625-12629, 2018 Nov 30.
Article
in English
| MEDLINE | ID: mdl-32232122