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1.
Structure-activity relationship of dibenzylideneacetone analogs against the neglected disease pathogen, Trypanosoma brucei.
Bioorg Med Chem Lett
; 81: 129123, 2023 02 01.
Article
in English
| MEDLINE | ID: mdl-36608774
2.
Targeting the Grb2 cSH3 domain: Design, synthesis and biological evaluation of the first series of modulators.
Bioorg Chem
; 138: 106607, 2023 09.
Article
in English
| MEDLINE | ID: mdl-37210829
3.
Emerging Direct Targeting ß-Catenin Agents.
Molecules
; 27(22)2022 Nov 10.
Article
in English
| MEDLINE | ID: mdl-36431838
4.
Emerging Therapeutic Agents for Colorectal Cancer.
Molecules
; 26(24)2021 Dec 09.
Article
in English
| MEDLINE | ID: mdl-34946546
5.
Modeling Epac1 interactions with the allosteric inhibitor AM-001 by co-solvent molecular dynamics.
J Comput Aided Mol Des
; 34(11): 1171-1179, 2020 11.
Article
in English
| MEDLINE | ID: mdl-32700175
6.
TRPA1 channels as targets for resveratrol and related stilbenoids.
Bioorg Med Chem Lett
; 26(3): 899-902, 2016 Feb 01.
Article
in English
| MEDLINE | ID: mdl-26750258
7.
Arylboronic acids as dual-action FAAH and TRPV1 ligands.
Bioorg Med Chem Lett
; 26(5): 1401-5, 2016 Mar 01.
Article
in English
| MEDLINE | ID: mdl-26850005
8.
Effect of acyclic monoterpene alcohols and their derivatives on TRP channels.
Bioorg Med Chem Lett
; 24(23): 5507-11, 2014 Dec 01.
Article
in English
| MEDLINE | ID: mdl-25455494
9.
3-Ylidenephthalides as a new class of transient receptor potential channel TRPA1 and TRPM8 modulators.
Bioorg Med Chem Lett
; 23(20): 5614-8, 2013 Oct 15.
Article
in English
| MEDLINE | ID: mdl-23993334
10.
Tetrahydro-ß-carboline derivatives targeting fatty acid amide hydrolase (FAAH) and transient receptor potential (TRP) channels.
Bioorg Med Chem Lett
; 23(1): 138-42, 2013 Jan 01.
Article
in English
| MEDLINE | ID: mdl-23206861
11.
RS6077 induces mitotic arrest and selectively activates cell death in human cancer cell lines and in a lymphoma tumor in vivo.
Eur J Med Chem
; 246: 114997, 2023 Jan 15.
Article
in English
| MEDLINE | ID: mdl-36502578
12.
Novel N-(Heterocyclylphenyl)benzensulfonamide Sharing an Unreported Binding Site with T-Cell Factor 4 at the ß-Catenin Armadillo Repeats Domain as an Anticancer Agent.
ACS Pharmacol Transl Sci
; 6(7): 1087-1103, 2023 Jul 14.
Article
in English
| MEDLINE | ID: mdl-37470018
13.
4-(3-Phenyl-4-(3,4,5-trimethoxybenzoyl)-1H-pyrrol-1-yl)benzenesulfonamide, a Novel Carbonic Anhydrase and Wnt/ß-Catenin Signaling Pathway Dual-Targeting Inhibitor with Potent Activity against Multidrug Resistant Cancer Cells.
J Med Chem
; 66(21): 14824-14842, 2023 11 09.
Article
in English
| MEDLINE | ID: mdl-37902628
14.
Synthesis and biological evaluation of [6]-gingerol analogues as transient receptor potential channel TRPV1 and TRPA1 modulators.
Bioorg Med Chem Lett
; 22(4): 1674-7, 2012 Feb 15.
Article
in English
| MEDLINE | ID: mdl-22257892
15.
Modulation of thermo-transient receptor potential (thermo-TRP) channels by thymol-based compounds.
Bioorg Med Chem Lett
; 22(10): 3535-9, 2012 May 15.
Article
in English
| MEDLINE | ID: mdl-22503249
16.
Discovery of novel human lactate dehydrogenase inhibitors: Structure-based virtual screening studies and biological assessment.
Eur J Med Chem
; 240: 114605, 2022 Oct 05.
Article
in English
| MEDLINE | ID: mdl-35868126
17.
Induction of Ferroptosis in Glioblastoma and Ovarian Cancers by a New Pyrrole Tubulin Assembly Inhibitor.
J Med Chem
; 65(23): 15805-15818, 2022 12 08.
Article
in English
| MEDLINE | ID: mdl-36395526
18.
Discovery of a Novel Class of Norovirus Inhibitors with High Barrier of Resistance.
Pharmaceuticals (Basel)
; 14(10)2021 Sep 30.
Article
in English
| MEDLINE | ID: mdl-34681230
19.
Targeting PDZ domains as potential treatment for viral infections, neurodegeneration and cancer.
Biol Direct
; 16(1): 15, 2021 10 12.
Article
in English
| MEDLINE | ID: mdl-34641953
20.
CXCR4 antagonism sensitizes cancer cells to novel indole-based MDM2/4 inhibitors in glioblastoma multiforme.
Eur J Pharmacol
; 897: 173936, 2021 Apr 15.
Article
in English
| MEDLINE | ID: mdl-33581134