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1.
Inhibition of the C1s Protease and the Classical Complement Pathway by 6-(4-Phenylpiperazin-1-yl)Pyridine-3-Carboximidamide and Chemical Analogs.
J Immunol
; 212(4): 689-701, 2024 Feb 15.
Article
in English
| MEDLINE | ID: mdl-38149922
2.
International Union of Basic and Clinical Pharmacology CXIII: Nuclear Receptor Superfamily-Update 2023.
Pharmacol Rev
; 75(6): 1233-1318, 2023 Nov.
Article
in English
| MEDLINE | ID: mdl-37586884
3.
Novel Pan-ERR Agonists Ameliorate Heart Failure Through Enhancing Cardiac Fatty Acid Metabolism and Mitochondrial Function.
Circulation
; 149(3): 227-250, 2024 01 16.
Article
in English
| MEDLINE | ID: mdl-37961903
4.
A Synthetic ERR Agonist Alleviates Metabolic Syndrome.
J Pharmacol Exp Ther
; 388(2): 232-240, 2024 01 17.
Article
in English
| MEDLINE | ID: mdl-37739806
5.
Estrogen-Related Receptor Agonism Reverses Mitochondrial Dysfunction and Inflammation in the Aging Kidney.
Am J Pathol
; 193(12): 1969-1987, 2023 12.
Article
in English
| MEDLINE | ID: mdl-37717940
6.
Identification and structure-activity relationships for a series of N, N-disubstituted 2-aminobenzothiazoles as potent inhibitors of S. aureus.
Bioorg Med Chem Lett
; 89: 129301, 2023 06 01.
Article
in English
| MEDLINE | ID: mdl-37094726
7.
Multidrug Efflux Pumps and the Two-Faced Janus of Substrates and Inhibitors.
Acc Chem Res
; 54(4): 930-939, 2021 02 16.
Article
in English
| MEDLINE | ID: mdl-33539084
8.
Sphingosine-1-phosphate receptor 1 activation in astrocytes contributes to neuropathic pain.
Proc Natl Acad Sci U S A
; 116(21): 10557-10562, 2019 05 21.
Article
in English
| MEDLINE | ID: mdl-31068460
9.
GPR183-Oxysterol Axis in Spinal Cord Contributes to Neuropathic Pain.
J Pharmacol Exp Ther
; 375(2): 367-375, 2020 11.
Article
in English
| MEDLINE | ID: mdl-32913007
10.
Machine Learning Algorithm Identifies an Antibiotic Vocabulary for Permeating Gram-Negative Bacteria.
J Chem Inf Model
; 60(6): 2838-2847, 2020 06 22.
Article
in English
| MEDLINE | ID: mdl-32453589
11.
Identification of C3b-Binding Small-Molecule Complement Inhibitors Using Cheminformatics.
J Immunol
; 198(9): 3705-3718, 2017 05 01.
Article
in English
| MEDLINE | ID: mdl-28298523
12.
AdeIJK Pump-Specific Inhibitors Effective against Multidrug Resistant Acinetobacter baumannii.
ACS Infect Dis
; 2024 May 24.
Article
in English
| MEDLINE | ID: mdl-38787939
13.
Predicting permeation of compounds across the outer membrane of P. aeruginosa using molecular descriptors.
Commun Chem
; 7(1): 84, 2024 Apr 12.
Article
in English
| MEDLINE | ID: mdl-38609430
14.
Development and pharmacological evaluation of a new chemical series of potent pan-ERR agonists, identification of SLU-PP-915.
Eur J Med Chem
; 258: 115582, 2023 Oct 05.
Article
in English
| MEDLINE | ID: mdl-37421886
15.
Synthetic ERRα/ß/γ Agonist Induces an ERRα-Dependent Acute Aerobic Exercise Response and Enhances Exercise Capacity.
ACS Chem Biol
; 18(4): 756-771, 2023 04 21.
Article
in English
| MEDLINE | ID: mdl-36988910
16.
Analysis of Orthogonal Efflux and Permeation Properties of Compounds Leads to the Discovery of New Efflux Pump Inhibitors.
ACS Infect Dis
; 8(10): 2149-2160, 2022 10 14.
Article
in English
| MEDLINE | ID: mdl-36070489
17.
Structural basis of synthetic agonist activation of the nuclear receptor REV-ERB.
Nat Commun
; 13(1): 7131, 2022 11 21.
Article
in English
| MEDLINE | ID: mdl-36414641
18.
Investigation of the pyrazinones as PDE5 inhibitors: evaluation of regioisomeric projections into the solvent region.
Bioorg Med Chem Lett
; 21(21): 6348-52, 2011 Nov 01.
Article
in English
| MEDLINE | ID: mdl-21955943
19.
Design, synthesis and activity of a potent, selective series of N-aryl pyridinone inhibitors of p38 kinase.
Bioorg Med Chem Lett
; 21(13): 4059-65, 2011 Jul 01.
Article
in English
| MEDLINE | ID: mdl-21640588
20.
Discovery of PH-797804, a highly selective and potent inhibitor of p38 MAP kinase.
Bioorg Med Chem Lett
; 21(13): 4066-71, 2011 Jul 01.
Article
in English
| MEDLINE | ID: mdl-21641211