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1.
Quantitative MS-Based Proteomics: Comparing the MCF-7 Cellular Response to Hypoxia and a 2-Oxoglutarate Analogue.
Chembiochem
; 21(11): 1647-1655, 2020 06 02.
Article
in English
| MEDLINE | ID: mdl-31919953
2.
Tuning the Transcriptional Response to Hypoxia by Inhibiting Hypoxia-inducible Factor (HIF) Prolyl and Asparaginyl Hydroxylases.
J Biol Chem
; 291(39): 20661-73, 2016 09 23.
Article
in English
| MEDLINE | ID: mdl-27502280
3.
Dual-action inhibitors of HIF prolyl hydroxylases that induce binding of a second iron ion.
Org Biomol Chem
; 11(5): 732-745, 2013 Feb 07.
Article
in English
| MEDLINE | ID: mdl-23151668
4.
Assays to Study Hypoxia-Inducible Factor Prolyl Hydroxylase Domain 2 (PHD2), a Key Human Oxygen Sensing Protein.
Methods Mol Biol
; 2648: 187-206, 2023.
Article
in English
| MEDLINE | ID: mdl-37039992
5.
Overview of the multifaceted resistances toward EGFR-TKIs and new chemotherapeutic strategies in non-small cell lung cancer.
Biochem Pharmacol
; 205: 115262, 2022 11.
Article
in English
| MEDLINE | ID: mdl-36191627
6.
NUB1 and FAT10 Proteins as Potential Novel Biomarkers in Cancer: A Translational Perspective.
Cells
; 10(9)2021 08 24.
Article
in English
| MEDLINE | ID: mdl-34571823
7.
Dynamic combinatorial chemistry employing boronic acids/boronate esters leads to potent oxygenase inhibitors.
Angew Chem Int Ed Engl
; 51(27): 6672-5, 2012 Jul 02.
Article
in English
| MEDLINE | ID: mdl-22639232
8.
Linking of 2-oxoglutarate and substrate binding sites enables potent and highly selective inhibition of JmjC histone demethylases.
Angew Chem Int Ed Engl
; 51(7): 1631-4, 2012 Feb 13.
Article
in English
| MEDLINE | ID: mdl-22241642
9.
Pharmacological targeting of the HIF hydroxylases--A new field in medicine development.
Mol Aspects Med
; 47-48: 54-75, 2016.
Article
in English
| MEDLINE | ID: mdl-26791432
10.
An experimentally validated network of nine haematopoietic transcription factors reveals mechanisms of cell state stability.
Elife
; 5: e11469, 2016 Feb 22.
Article
in English
| MEDLINE | ID: mdl-26901438
11.
Potent and Selective Triazole-Based Inhibitors of the Hypoxia-Inducible Factor Prolyl-Hydroxylases with Activity in the Murine Brain.
PLoS One
; 10(7): e0132004, 2015.
Article
in English
| MEDLINE | ID: mdl-26147748
12.
Inhibition of the HIF1α-p300 interaction by quinone- and indandione-mediated ejection of structural Zn(II).
Eur J Med Chem
; 94: 509-16, 2015 Apr 13.
Article
in English
| MEDLINE | ID: mdl-25023609
13.
Non-enzymatic chemistry enables 2-hydroxyglutarate-mediated activation of 2-oxoglutarate oxygenases.
Nat Commun
; 5: 3423, 2014 Mar 05.
Article
in English
| MEDLINE | ID: mdl-24594748
14.
A cell-permeable ester derivative of the JmjC histone demethylase inhibitor IOX1.
ChemMedChem
; 9(3): 566-71, 2014 Mar.
Article
in English
| MEDLINE | ID: mdl-24504543
15.
Selective small molecule probes for the hypoxia inducible factor (HIF) prolyl hydroxylases.
ACS Chem Biol
; 8(7): 1488-96, 2013 Jul 19.
Article
in English
| MEDLINE | ID: mdl-23683440
16.
5-Carboxy-8-hydroxyquinoline is a Broad Spectrum 2-Oxoglutarate Oxygenase Inhibitor which Causes Iron Translocation.
Chem Sci
; 4(8): 3110-3117, 2013 Aug 01.
Article
in English
| MEDLINE | ID: mdl-26682036
17.
Plant growth regulator daminozide is a selective inhibitor of human KDM2/7 histone demethylases.
J Med Chem
; 55(14): 6639-43, 2012 Jul 26.
Article
in English
| MEDLINE | ID: mdl-22724510
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