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1.
Stack-VTP: prediction of vesicle transport proteins based on stacked ensemble classifier and evolutionary information.
BMC Bioinformatics
; 24(1): 137, 2023 Apr 07.
Article
in English
| MEDLINE | ID: mdl-37029385
2.
Design, Synthesis and Evaluation of Fluorescent Properties of Benzothiazole Derivatives.
Chemphyschem
; 24(17): e202300159, 2023 09 01.
Article
in English
| MEDLINE | ID: mdl-37349282
3.
Exploration of novel four-membered-heterocycle constructed peptidyl proteasome inhibitors with improved metabolic stability for cancer treatment.
Bioorg Chem
; 138: 106626, 2023 09.
Article
in English
| MEDLINE | ID: mdl-37295239
4.
Synthesis and Biological Evaluation of 3-Amino-4,4-Dimethyl Lithocholic Acid Derivatives as Novel, Selective, and Cellularly Active Allosteric SHP1 Activators.
Molecules
; 28(6)2023 Mar 08.
Article
in English
| MEDLINE | ID: mdl-36985458
5.
Theoretical study and application of 2-phenyl-1,3,4-thiadiazole derivatives with optical and inhibitory activity against SHP1.
Phys Chem Chem Phys
; 24(2): 861-874, 2022 Jan 04.
Article
in English
| MEDLINE | ID: mdl-34908073
6.
Synthesis and Biochemical Evaluation of 8H-Indeno[1,2-d]thiazole Derivatives as Novel SARS-CoV-2 3CL Protease Inhibitors.
Molecules
; 27(10)2022 May 23.
Article
in English
| MEDLINE | ID: mdl-35630836
7.
Synthesis and biological evaluation of 2,5-diaryl-1,3,4-oxadiazole derivatives as novel Src homology 2 domain-containing protein tyrosine phosphatase 2 (SHP2) inhibitors.
Bioorg Chem
; 116: 105384, 2021 11.
Article
in English
| MEDLINE | ID: mdl-34601294
8.
Synthesis and biological evaluation of heterocyclic bis-aryl amides as novel Src homology 2 domain containing protein tyrosine phosphatase-2 (SHP2) inhibitors.
Bioorg Med Chem Lett
; 30(11): 127170, 2020 06 01.
Article
in English
| MEDLINE | ID: mdl-32273218
9.
Efficient synthesis, biological evaluation, and docking study of isatin based derivatives as caspase inhibitors.
J Enzyme Inhib Med Chem
; 35(1): 1674-1684, 2020 Dec.
Article
in English
| MEDLINE | ID: mdl-32842789
10.
Discovery of 1,3-diphenyl-1H-pyrazole derivatives containing rhodanine-3-alkanoic acid groups as potential PTP1B inhibitors.
Bioorg Med Chem Lett
; 29(10): 1187-1193, 2019 05 15.
Article
in English
| MEDLINE | ID: mdl-30910462
11.
Synthesis and biological evaluation of 3-aryl-4-indolyl-maleimides as potent mutant isocitrate dehydrogenase-1 inhibitors.
Bioorg Med Chem
; 27(4): 589-603, 2019 02 15.
Article
in English
| MEDLINE | ID: mdl-30600148
12.
3-(7-Azaindolyl)-4-indolylmaleimides as a novel class of mutant isocitrate dehydrogenase-1 inhibitors: Design, synthesis, and biological evaluation.
Arch Pharm (Weinheim)
; 351(10): e1800039, 2018 Oct.
Article
in English
| MEDLINE | ID: mdl-30113716
13.
Tim3/galectin-9 alleviates the inflammation of TAO patients via suppressing Akt/NF-kB signaling pathway.
Biochem Biophys Res Commun
; 491(4): 966-972, 2017 09 30.
Article
in English
| MEDLINE | ID: mdl-28756232
14.
Discovery of core-structurally novel PTP1B inhibitors with specific selectivity containing oxindole-fused spirotetrahydrofurochroman by one-pot reaction.
Bioorg Med Chem Lett
; 27(4): 1105-1108, 2017 02 15.
Article
in English
| MEDLINE | ID: mdl-28111140
15.
Benzo[c][1,2,5]thiadiazole derivatives: A new class of potent Src homology-2 domain containing protein tyrosine phosphatase-2 (SHP2) inhibitors.
Bioorg Med Chem Lett
; 27(23): 5154-5157, 2017 12 01.
Article
in English
| MEDLINE | ID: mdl-29100798
16.
Synthesis and biological evaluation of novel 4,5-bisindolyl-1,2,4-triazol-3-ones as glycogen synthase kinase-3ß inhibitors and neuroprotective agents.
Pharmazie
; 72(12): 707-713, 2017 Dec 01.
Article
in English
| MEDLINE | ID: mdl-29441954
17.
Compartmentalized gene regulatory network of the pathogenic fungus Fusarium graminearum.
New Phytol
; 211(2): 527-41, 2016 07.
Article
in English
| MEDLINE | ID: mdl-26990214
18.
Design, synthesis and in vitro activity of phidianidine B derivatives as novel PTP1B inhibitors with specific selectivity.
Bioorg Med Chem Lett
; 26(3): 778-781, 2016 Feb 01.
Article
in English
| MEDLINE | ID: mdl-26774579
19.
Design, synthesis and biological evaluation of novel non-covalent piperidine-containing peptidyl proteasome inhibitors.
Bioorg Med Chem
; 24(23): 6206-6214, 2016 12 01.
Article
in English
| MEDLINE | ID: mdl-27765408
20.
Curcusone D, a novel ubiquitin-proteasome pathway inhibitor via ROS-induced DUB inhibition, is synergistic with bortezomib against multiple myeloma cell growth.
Biochim Biophys Acta
; 1840(6): 2004-13, 2014 Jun.
Article
in English
| MEDLINE | ID: mdl-24534329