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1.
Coupling the Antimalarial Cell Penetrating Peptide TP10 to Classical Antimalarial Drugs Primaquine and Chloroquine Produces Strongly Hemolytic Conjugates.
Molecules
; 24(24)2019 Dec 12.
Article
in English
| MEDLINE | ID: mdl-31842498
2.
Cryptosporidium and Toxoplasma Parasites Are Inhibited by a Benzoxaborole Targeting Leucyl-tRNA Synthetase.
Antimicrob Agents Chemother
; 60(10): 5817-27, 2016 10.
Article
in English
| MEDLINE | ID: mdl-27431220
3.
Antimalarial Benzoxaboroles Target Plasmodium falciparum Leucyl-tRNA Synthetase.
Antimicrob Agents Chemother
; 60(8): 4886-95, 2016 08.
Article
in English
| MEDLINE | ID: mdl-27270277
4.
Novel squaramides with in vitro liver stage antiplasmodial activity.
Bioorg Med Chem
; 24(8): 1786-92, 2016 Apr 15.
Article
in English
| MEDLINE | ID: mdl-26968650
5.
Chemical genetics of Plasmodium falciparum.
Nature
; 465(7296): 311-5, 2010 May 20.
Article
in English
| MEDLINE | ID: mdl-20485428
6.
Impact of antimalarial treatment and chemoprevention on the drug sensitivity of malaria parasites isolated from ugandan children.
Antimicrob Agents Chemother
; 59(6): 3018-30, 2015.
Article
in English
| MEDLINE | ID: mdl-25753626
7.
Tetrafluorophenoxymethyl ketone cruzain inhibitors with improved pharmacokinetic properties as therapeutic leads for Chagas' disease.
Bioorg Med Chem Lett
; 25(21): 4834-4837, 2015 Nov 01.
Article
in English
| MEDLINE | ID: mdl-26144347
8.
N10,N11-di-alkylamine indolo[3,2-b]quinolines as hemozoin inhibitors: design, synthesis and antiplasmodial activity.
Bioorg Med Chem
; 23(7): 1530-9, 2015 Apr 01.
Article
in English
| MEDLINE | ID: mdl-25725608
9.
Hsp90 inhibitors as new leads to target parasitic diarrheal diseases.
Antimicrob Agents Chemother
; 58(7): 4138-44, 2014 Jul.
Article
in English
| MEDLINE | ID: mdl-24820073
10.
1H-1,2,3-Triazole-tethered isatin-7-chloroquinoline and 3-hydroxy-indole-7-chloroquinoline conjugates: synthesis and antimalarial evaluation.
Bioorg Med Chem Lett
; 24(3): 756-9, 2014 Feb 01.
Article
in English
| MEDLINE | ID: mdl-24424135
11.
Synthesis, biological evaluation, hydration site thermodynamics, and chemical reactivity analysis of α-keto substituted peptidomimetics for the inhibition of Plasmodium falciparum.
Bioorg Med Chem Lett
; 24(5): 1274-9, 2014 Mar 01.
Article
in English
| MEDLINE | ID: mdl-24507921
12.
A reprofiled drug, auranofin, is effective against metronidazole-resistant Giardia lamblia.
Antimicrob Agents Chemother
; 57(5): 2029-35, 2013 May.
Article
in English
| MEDLINE | ID: mdl-23403423
13.
In vitro and in vivo antimalarial efficacies of optimized tetracyclines.
Antimicrob Agents Chemother
; 57(7): 3131-6, 2013 Jul.
Article
in English
| MEDLINE | ID: mdl-23629719
14.
In vitro efficiency of 9-(N-cinnamoylbutyl)aminoacridines against blood- and liver-stage malaria parasites.
Bioorg Med Chem Lett
; 23(3): 610-3, 2013 Feb 01.
Article
in English
| MEDLINE | ID: mdl-23290049
15.
Novel anti-plasmodial hits identified by virtual screening of the ZINC database.
J Comput Aided Mol Des
; 27(10): 859-71, 2013 Oct.
Article
in English
| MEDLINE | ID: mdl-24158745
16.
Tetrazole-based deoxyamodiaquines: synthesis, ADME/PK profiling and pharmacological evaluation as potential antimalarial agents.
Bioorg Med Chem
; 21(17): 4904-13, 2013 Sep 01.
Article
in English
| MEDLINE | ID: mdl-23896611
17.
Chemical-biological characterization of a cruzain inhibitor reveals a second target and a mammalian off-target.
Beilstein J Org Chem
; 9: 15-25, 2013.
Article
in English
| MEDLINE | ID: mdl-23400640
18.
Artefenomel Regioisomer RLA-3107 Is a Promising Lead for the Discovery of Next-Generation Endoperoxide Antimalarials.
ACS Med Chem Lett
; 14(4): 493-498, 2023 Apr 13.
Article
in English
| MEDLINE | ID: mdl-37077383
19.
Novel potent metallocenes against liver stage malaria.
Antimicrob Agents Chemother
; 56(3): 1564-70, 2012 Mar.
Article
in English
| MEDLINE | ID: mdl-22155838
20.
Compounds from Sorindeia juglandifolia (Anacardiaceae) exhibit potent anti-plasmodial activities in vitro and in vivo.
Malar J
; 11: 382, 2012 Nov 21.
Article
in English
| MEDLINE | ID: mdl-23171238