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Synthesis and biological evaluation of a series of novel pyridinecarboxamides as potential multi-receptor antipsychotic drugs.
Xu, Mingshuo; Wang, Yu; Yang, Feipu; Wu, Chunhui; Wang, Zhen; Ye, Bin; Jiang, Xiangrui; Zhao, Qingjie; Li, Jianfeng; Liu, Yongjian; Zhang, Junchi; Tian, Guanghui; He, Yang; Shen, Jingshan; Jiang, Hualiang.
Affiliation
  • Xu M; CAS Key Laboratory for Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China; University of Chinese Academy of Sciences, No. 19A Yuquan Road, Beijing 100049, China.
  • Wang Y; CAS Key Laboratory for Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China.
  • Yang F; CAS Key Laboratory for Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China.
  • Wu C; Topharman Shanghai Co., Ltd, 1088 Chuansha Road, Shanghai 201209, China.
  • Wang Z; CAS Key Laboratory for Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China.
  • Ye B; Topharman Shanghai Co., Ltd, 1088 Chuansha Road, Shanghai 201209, China.
  • Jiang X; CAS Key Laboratory for Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China.
  • Zhao Q; CAS Key Laboratory for Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China.
  • Li J; CAS Key Laboratory for Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China.
  • Liu Y; Topharman Shanghai Co., Ltd, 1088 Chuansha Road, Shanghai 201209, China.
  • Zhang J; CAS Key Laboratory for Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China.
  • Tian G; Topharman Shanghai Co., Ltd, 1088 Chuansha Road, Shanghai 201209, China.
  • He Y; CAS Key Laboratory for Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China. Electronic address: heyang@simm.ac.cn.
  • Shen J; CAS Key Laboratory for Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China. Electronic address: shenjingshan@simm.ac.cn.
  • Jiang H; CAS Key Laboratory for Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China.
Bioorg Med Chem Lett ; 28(4): 606-611, 2018 02 15.
Article in En | MEDLINE | ID: mdl-29395980

Full text: 1 Database: MEDLINE Main subject: Picolinic Acids / Antipsychotic Agents Limits: Animals / Humans / Male Language: En Year: 2018 Type: Article

Full text: 1 Database: MEDLINE Main subject: Picolinic Acids / Antipsychotic Agents Limits: Animals / Humans / Male Language: En Year: 2018 Type: Article