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Investigation of biaryl heterocycles as inhibitors of Wee1 kinase.
Mastracchio, Anthony; Lai, Chunqiu; Torrent, Maricel; Bromberg, Kenneth; Buchanan, Fritz G; Ferguson, Debra; Bontcheva, Velitchka; Johnson, Eric F; Lasko, Loren; Maag, David; Shoemaker, Alexander R; Penning, Thomas D.
Affiliation
  • Mastracchio A; Cancer Research, Discovery, Global Pharmaceutical Research and Development, AbbVie, 1 North Waukegan Road, North Chicago, IL 60064, United States. Electronic address: anthony.mastracchio@abbvie.com.
  • Lai C; Cancer Research, Discovery, Global Pharmaceutical Research and Development, AbbVie, 1 North Waukegan Road, North Chicago, IL 60064, United States.
  • Torrent M; Molecular Modeling, Structural Biology, Discovery, Global Pharmaceutical Research and Development, AbbVie, 1 North Waukegan Road, North Chicago, IL 60064, United States.
  • Bromberg K; Cancer Research, Discovery, Global Pharmaceutical Research and Development, AbbVie, 1 North Waukegan Road, North Chicago, IL 60064, United States.
  • Buchanan FG; Cancer Research, Discovery, Global Pharmaceutical Research and Development, AbbVie, 1 North Waukegan Road, North Chicago, IL 60064, United States.
  • Ferguson D; Cancer Research, Discovery, Global Pharmaceutical Research and Development, AbbVie, 1 North Waukegan Road, North Chicago, IL 60064, United States.
  • Bontcheva V; Cancer Research, Discovery, Global Pharmaceutical Research and Development, AbbVie, 1 North Waukegan Road, North Chicago, IL 60064, United States.
  • Johnson EF; Cancer Research, Discovery, Global Pharmaceutical Research and Development, AbbVie, 1 North Waukegan Road, North Chicago, IL 60064, United States.
  • Lasko L; Cancer Research, Discovery, Global Pharmaceutical Research and Development, AbbVie, 1 North Waukegan Road, North Chicago, IL 60064, United States.
  • Maag D; Cancer Research, Discovery, Global Pharmaceutical Research and Development, AbbVie, 1 North Waukegan Road, North Chicago, IL 60064, United States.
  • Shoemaker AR; Cancer Research, Discovery, Global Pharmaceutical Research and Development, AbbVie, 1 North Waukegan Road, North Chicago, IL 60064, United States.
  • Penning TD; Cancer Research, Discovery, Global Pharmaceutical Research and Development, AbbVie, 1 North Waukegan Road, North Chicago, IL 60064, United States.
Bioorg Med Chem Lett ; 29(12): 1481-1486, 2019 06 15.
Article in En | MEDLINE | ID: mdl-31014911

Full text: 1 Database: MEDLINE Main subject: Protein-Tyrosine Kinases / Cell Cycle Proteins / Heterocyclic Compounds Limits: Humans Language: En Year: 2019 Type: Article

Full text: 1 Database: MEDLINE Main subject: Protein-Tyrosine Kinases / Cell Cycle Proteins / Heterocyclic Compounds Limits: Humans Language: En Year: 2019 Type: Article