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Identification and Characterization of Dual Inhibitors of the USP25/28 Deubiquitinating Enzyme Subfamily.
Wrigley, Jonathan D; Gavory, Gerald; Simpson, Iain; Preston, Marian; Plant, Helen; Bradley, Jenna; Goeppert, Anne U; Rozycka, Ewelina; Davies, Gareth; Walsh, Jarrod; Valentine, Andrea; McClelland, Keeva; Odrzywol, Krzysztofa Ewa; Renshaw, Jonathan; Boros, Joanna; Tart, Jonathan; Leach, Lindsey; Nowak, Thorsten; Ward, Richard A; Harrison, Timothy; Andrews, David M.
Afiliación
  • Wrigley JD; Discovery Sciences, IMED Biotech Unit, AstraZeneca , Cambridge, United Kingdom.
  • Gavory G; Almac Discovery Ltd. , Centre for Precision Therapeutics, 97 Lisburn Road, Belfast, BT9 7AE, United Kingdom.
  • Simpson I; Oncology, IMED Biotech Unit, AstraZeneca , Cambridge, United Kingdom.
  • Preston M; Discovery Sciences, IMED Biotech Unit, AstraZeneca , Cambridge, United Kingdom.
  • Plant H; Discovery Sciences, IMED Biotech Unit, AstraZeneca , Cambridge, United Kingdom.
  • Bradley J; Discovery Sciences, IMED Biotech Unit, AstraZeneca , Cambridge, United Kingdom.
  • Goeppert AU; Discovery Sciences, IMED Biotech Unit, AstraZeneca , Cambridge, United Kingdom.
  • Rozycka E; Almac Discovery Ltd. , Centre for Precision Therapeutics, 97 Lisburn Road, Belfast, BT9 7AE, United Kingdom.
  • Davies G; Discovery Sciences, IMED Biotech Unit, AstraZeneca , Cambridge, United Kingdom.
  • Walsh J; Discovery Sciences, IMED Biotech Unit, AstraZeneca , Cambridge, United Kingdom.
  • Valentine A; Almac Discovery Ltd. , Centre for Precision Therapeutics, 97 Lisburn Road, Belfast, BT9 7AE, United Kingdom.
  • McClelland K; Almac Discovery Ltd. , Centre for Precision Therapeutics, 97 Lisburn Road, Belfast, BT9 7AE, United Kingdom.
  • Odrzywol KE; Almac Discovery Ltd. , Centre for Precision Therapeutics, 97 Lisburn Road, Belfast, BT9 7AE, United Kingdom.
  • Renshaw J; Discovery Sciences, IMED Biotech Unit, AstraZeneca , Cambridge, United Kingdom.
  • Boros J; Discovery Sciences, IMED Biotech Unit, AstraZeneca , Cambridge, United Kingdom.
  • Tart J; Discovery Sciences, IMED Biotech Unit, AstraZeneca , Cambridge, United Kingdom.
  • Leach L; Discovery Sciences, IMED Biotech Unit, AstraZeneca , Cambridge, United Kingdom.
  • Nowak T; Oncology, IMED Biotech Unit, AstraZeneca , Cambridge, United Kingdom.
  • Ward RA; Oncology, IMED Biotech Unit, AstraZeneca , Cambridge, United Kingdom.
  • Harrison T; Almac Discovery Ltd. , Centre for Precision Therapeutics, 97 Lisburn Road, Belfast, BT9 7AE, United Kingdom.
  • Andrews DM; Oncology, IMED Biotech Unit, AstraZeneca , Cambridge, United Kingdom.
ACS Chem Biol ; 12(12): 3113-3125, 2017 12 15.
Article en En | MEDLINE | ID: mdl-29131570

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Ubiquitina Tiolesterasa / Inhibidores Enzimáticos / Antineoplásicos Tipo de estudio: Diagnostic_studies / Prognostic_studies Límite: Humans Idioma: En Año: 2017 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Ubiquitina Tiolesterasa / Inhibidores Enzimáticos / Antineoplásicos Tipo de estudio: Diagnostic_studies / Prognostic_studies Límite: Humans Idioma: En Año: 2017 Tipo del documento: Article