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Pharmacological Characterization of Aprocitentan, a Dual Endothelin Receptor Antagonist, Alone and in Combination with Blockers of the Renin Angiotensin System, in Two Models of Experimental Hypertension.
Trensz, Frederic; Bortolamiol, Céline; Kramberg, Markus; Wanner, Daniel; Hadana, Hakim; Rey, Markus; Strasser, Daniel S; Delahaye, Stéphane; Hess, Patrick; Vezzali, Enrico; Mentzel, Ulrich; Ménard, Joël; Clozel, Martine; Iglarz, Marc.
Afiliación
  • Trensz F; Drug Discovery Department, Idorsia Pharmaceuticals Ltd., Allschwil, Switzerland.
  • Bortolamiol C; Drug Discovery Department, Idorsia Pharmaceuticals Ltd., Allschwil, Switzerland.
  • Kramberg M; Drug Discovery Department, Idorsia Pharmaceuticals Ltd., Allschwil, Switzerland.
  • Wanner D; Drug Discovery Department, Idorsia Pharmaceuticals Ltd., Allschwil, Switzerland.
  • Hadana H; Drug Discovery Department, Idorsia Pharmaceuticals Ltd., Allschwil, Switzerland.
  • Rey M; Drug Discovery Department, Idorsia Pharmaceuticals Ltd., Allschwil, Switzerland.
  • Strasser DS; Drug Discovery Department, Idorsia Pharmaceuticals Ltd., Allschwil, Switzerland.
  • Delahaye S; Drug Discovery Department, Idorsia Pharmaceuticals Ltd., Allschwil, Switzerland.
  • Hess P; Drug Discovery Department, Idorsia Pharmaceuticals Ltd., Allschwil, Switzerland.
  • Vezzali E; Drug Discovery Department, Idorsia Pharmaceuticals Ltd., Allschwil, Switzerland.
  • Mentzel U; Drug Discovery Department, Idorsia Pharmaceuticals Ltd., Allschwil, Switzerland.
  • Ménard J; Drug Discovery Department, Idorsia Pharmaceuticals Ltd., Allschwil, Switzerland.
  • Clozel M; Drug Discovery Department, Idorsia Pharmaceuticals Ltd., Allschwil, Switzerland.
  • Iglarz M; Drug Discovery Department, Idorsia Pharmaceuticals Ltd., Allschwil, Switzerland marc.iglarz@idorsia.com.
J Pharmacol Exp Ther ; 368(3): 462-473, 2019 03.
Article en En | MEDLINE | ID: mdl-30622171

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Pirimidinas / Sistema Renina-Angiotensina / Sulfonamidas / Antagonistas de los Receptores de Endotelina / Hipertensión / Antihipertensivos Tipo de estudio: Prognostic_studies Límite: Animals Idioma: En Año: 2019 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Pirimidinas / Sistema Renina-Angiotensina / Sulfonamidas / Antagonistas de los Receptores de Endotelina / Hipertensión / Antihipertensivos Tipo de estudio: Prognostic_studies Límite: Animals Idioma: En Año: 2019 Tipo del documento: Article