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Asymmetric Synthesis of a 5,6,7,8-Tetrahydro-1,6-naphthyridine Scaffold Leading to Potent Retinoid-Related Orphan Receptor γt Inverse Agonist TAK-828F.
Tsuruoka, Ryoji; Yoshikawa, Naoki; Konishi, Takahiro; Yamano, Mitsuhisa.
Afiliación
  • Tsuruoka R; Process Chemistry, Pharmaceutical Sciences, Takeda Pharmaceutical Company Limited, 17-85 Jusohonmachi 2-Chome, Yodogawa-ku, Osaka 532-8686, Japan.
  • Yoshikawa N; Process Chemistry, Pharmaceutical Sciences, Takeda Pharmaceutical Company Limited, 17-85 Jusohonmachi 2-Chome, Yodogawa-ku, Osaka 532-8686, Japan.
  • Konishi T; Process Chemistry, Pharmaceutical Sciences, Takeda Pharmaceutical Company Limited, 17-85 Jusohonmachi 2-Chome, Yodogawa-ku, Osaka 532-8686, Japan.
  • Yamano M; Process Chemistry, Pharmaceutical Sciences, Takeda Pharmaceutical Company Limited, 17-85 Jusohonmachi 2-Chome, Yodogawa-ku, Osaka 532-8686, Japan.
J Org Chem ; 85(16): 10797-10805, 2020 08 21.
Article en En | MEDLINE | ID: mdl-32701287

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Miembro 3 del Grupo F de la Subfamilia 1 de Receptores Nucleares / Naftiridinas Idioma: En Año: 2020 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Miembro 3 del Grupo F de la Subfamilia 1 de Receptores Nucleares / Naftiridinas Idioma: En Año: 2020 Tipo del documento: Article