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Optimization of linear and cyclic peptide inhibitors of KEAP1-NRF2 protein-protein interaction.
Colarusso, Stefania; De Simone, Daniele; Frattarelli, Tommaso; Andreini, Matteo; Cerretani, Mauro; Missineo, Antonino; Moretti, Daniele; Tambone, Sara; Kempf, Georg; Augustin, Martin; Steinbacher, Stefan; Munoz-Sanjuan, Ignacio; Park, Larry; Summa, Vincenzo; Tomei, Licia; Bresciani, Alberto; Dominguez, Celia; Toledo-Sherman, Leticia; Bianchi, Elisabetta.
Afiliación
  • Colarusso S; Department of Drug Discovery, IRBM Spa, Via Pontina km 30.600, 00071 Pomezia, Rome, Italy. Electronic address: s.colarusso@irbm.com.
  • De Simone D; Department of Drug Discovery, IRBM Spa, Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
  • Frattarelli T; Department of Drug Discovery, IRBM Spa, Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
  • Andreini M; Department of Drug Discovery, IRBM Spa, Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
  • Cerretani M; Translational & Discovery Research, IRBM Spa, Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
  • Missineo A; Translational & Discovery Research, IRBM Spa, Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
  • Moretti D; Translational & Discovery Research, IRBM Spa, Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
  • Tambone S; Translational & Discovery Research, IRBM Spa, Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
  • Kempf G; Proteros Biostructures GmbH, Bunsenstraße 7 a, 82152 Planegg, Germany.
  • Augustin M; Proteros Biostructures GmbH, Bunsenstraße 7 a, 82152 Planegg, Germany.
  • Steinbacher S; Proteros Biostructures GmbH, Bunsenstraße 7 a, 82152 Planegg, Germany.
  • Munoz-Sanjuan I; CHDI Management/CHDI Foundation, Los Angeles, CA, United States.
  • Park L; CHDI Management/CHDI Foundation, Los Angeles, CA, United States.
  • Summa V; Department of Drug Discovery, IRBM Spa, Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
  • Tomei L; Translational & Discovery Research, IRBM Spa, Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
  • Bresciani A; Translational & Discovery Research, IRBM Spa, Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
  • Dominguez C; CHDI Management/CHDI Foundation, Los Angeles, CA, United States. Electronic address: celia.dominguez@chdifoundation.org.
  • Toledo-Sherman L; Translational & Discovery Research, IRBM Spa, Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
  • Bianchi E; Department of Drug Discovery, IRBM Spa, Via Pontina km 30.600, 00071 Pomezia, Rome, Italy.
Bioorg Med Chem ; 28(21): 115738, 2020 11 01.
Article en En | MEDLINE | ID: mdl-33065433

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Péptidos / Péptidos Cíclicos / Factor 2 Relacionado con NF-E2 / Proteína 1 Asociada A ECH Tipo Kelch Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Año: 2020 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Péptidos / Péptidos Cíclicos / Factor 2 Relacionado con NF-E2 / Proteína 1 Asociada A ECH Tipo Kelch Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Año: 2020 Tipo del documento: Article