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In Vitro and In Vivo Pharmacological Characterization of a Novel TRPM8 Inhibitor Chemotype Identified by Small-Scale Preclinical Screening.
Iraci, Nunzio; Ostacolo, Carmine; Medina-Peris, Alicia; Ciaglia, Tania; Novoselov, Anton M; Altieri, Andrea; Cabañero, David; Fernandez-Carvajal, Asia; Campiglia, Pietro; Gomez-Monterrey, Isabel; Bertamino, Alessia; Kurkin, Alexander V.
Afiliación
  • Iraci N; Department of Chemical, Biological, Pharmaceutical and Environmental Sciences, University of Messina, Viale Ferdinando Stagno d'Alcontres 31, 98166 Messina, Italy.
  • Ostacolo C; Department of Pharmacy, University of Naples Federico II, Via D. Montesano 49, 80131 Naples, Italy.
  • Medina-Peris A; Instituto de Investigación, Desarrollo e Innovación en Biotecnología Sanitaria de Elche (IDiBE), Universidad Miguel Hernández de Elche, Avenida de la Universidad, 03202 Elche, Spain.
  • Ciaglia T; Department of Pharmacy, University of Salerno, Via G. Paolo II, 84084 Fisciano, Italy.
  • Novoselov AM; Department of Chemistry, Lomonosov Moscow State University, 1/3 Leninsky Gory, 119991 Moscow, Russia.
  • Altieri A; Department of Chemistry, Lomonosov Moscow State University, 1/3 Leninsky Gory, 119991 Moscow, Russia.
  • Cabañero D; EDASA Scientific srls, Via Stingi 37, 66050 San Salvo, Italy.
  • Fernandez-Carvajal A; Instituto de Investigación, Desarrollo e Innovación en Biotecnología Sanitaria de Elche (IDiBE), Universidad Miguel Hernández de Elche, Avenida de la Universidad, 03202 Elche, Spain.
  • Campiglia P; Instituto de Investigación, Desarrollo e Innovación en Biotecnología Sanitaria de Elche (IDiBE), Universidad Miguel Hernández de Elche, Avenida de la Universidad, 03202 Elche, Spain.
  • Gomez-Monterrey I; Department of Pharmacy, University of Salerno, Via G. Paolo II, 84084 Fisciano, Italy.
  • Bertamino A; Department of Pharmacy, University of Naples Federico II, Via D. Montesano 49, 80131 Naples, Italy.
  • Kurkin AV; Department of Pharmacy, University of Salerno, Via G. Paolo II, 84084 Fisciano, Italy.
Int J Mol Sci ; 23(4)2022 Feb 13.
Article en En | MEDLINE | ID: mdl-35216186

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Canales Catiónicos TRPM Tipo de estudio: Diagnostic_studies / Screening_studies Límite: Animals Idioma: En Año: 2022 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Canales Catiónicos TRPM Tipo de estudio: Diagnostic_studies / Screening_studies Límite: Animals Idioma: En Año: 2022 Tipo del documento: Article