1.
Bioorg Med Chem Lett
; 22(24): 7297-301, 2012 Dec 15.
Artículo
en Inglés
| MEDLINE
| ID: mdl-23159569
RESUMEN
We describe a novel 7-aminopyrazolo[1,5-a]pyrimidine (7-APP) derivative as a potent hepatitis C virus (HCV) inhibitor. A series of 7-APPs was synthesized and evaluated for inhibitory activity against HCV in different cell culture systems. The synthesis and preliminary structure-activity relationship study of 7-APP are reported.