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1.
Fitoterapia ; 145: 104613, 2020 Sep.
Artículo en Inglés | MEDLINE | ID: mdl-32407877

RESUMEN

Seven rare oxylipins, siegesbeckins A-G (1-7) representing further bioactive constituents different from the general terpenyl compounds found in Siegesbeckia species, have been obtained from the aerial parts of Siegesbeckia glabrescens. These isolates were identified to be a series of methyl 4-methylpentanoates incorporating fatty acid moieties of different chain lengths, based on spectroscopic techniques, and their absolute configurations were determined via chemical degradation and comparison of experimental and theoretically calculated ECD spectra. With respect to bioactivity, antibacterial, anti-inflammatory and cytotoxic properties of selected compounds were evaluated. Compounds 1 and 5 showed moderate antibacterial activity against two Gram-positive bacteria with MIC values of 4.3 µg/mL, while 3 showed no pronounced activity in these assays.


Asunto(s)
Antibacterianos/farmacología , Asteraceae/química , Oxilipinas/farmacología , Células A549 , Animales , Antibacterianos/aislamiento & purificación , Línea Celular Tumoral , China , Bacterias Grampositivas/efectos de los fármacos , Humanos , Ratones , Pruebas de Sensibilidad Microbiana , Estructura Molecular , Oxilipinas/aislamiento & purificación , Fitoquímicos/aislamiento & purificación , Fitoquímicos/farmacología , Componentes Aéreos de las Plantas/química , Células RAW 264.7
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