1.
Bioorg Med Chem Lett
; 17(22): 6066-9, 2007 Nov 15.
Artigo
em Inglês
| MEDLINE
| ID: mdl-17911022
RESUMO
In the course of our research program to develop novel muscarinic receptor antagonists for the treatment of COPD, new tropane carbamate derivatives were identified as potent anti-muscarinic agents. The synthesis, structure-activity relationships and pharmacological evaluation that led to the identification of compound 5o, are described.