1.
Bioorg Med Chem Lett
; 16(4): 845-9, 2006 Feb 15.
Artigo
em Inglês
| MEDLINE
| ID: mdl-16303301
RESUMO
We describe a series of 2,5 thiazole containing compounds, which are potent antagonists of the integrin alpha(v)beta3 and show selectivity relative to the other integrins, such as alpha(IIb)beta3 and alpha(v)beta6. These analogs were demonstrated to have high bioavailability relative to other relative heterocyclic analogs.