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Fluorescence-based assay for polyprenyl phosphate-GlcNAc-1-phosphate transferase (WecA) and identification of novel antimycobacterial WecA inhibitors.
Mitachi, Katsuhiko; Siricilla, Shajila; Yang, Dong; Kong, Ying; Skorupinska-Tudek, Karolina; Swiezewska, Ewa; Franzblau, Scott G; Kurosu, Michio.
Afiliación
  • Mitachi K; Department of Pharmaceutical Sciences, College of Pharmacy, University of Tennessee Health Science Center, 881 Madison Avenue, Memphis, TN 38163-0001, United States.
  • Siricilla S; Department of Pharmaceutical Sciences, College of Pharmacy, University of Tennessee Health Science Center, 881 Madison Avenue, Memphis, TN 38163-0001, United States.
  • Yang D; Department of Microbiology, Immunology & Biochemistry, University of Tennessee Health Science Center, 858 Madison Avenue, Memphis, TN 38163-0001, United Sates.
  • Kong Y; Department of Microbiology, Immunology & Biochemistry, University of Tennessee Health Science Center, 858 Madison Avenue, Memphis, TN 38163-0001, United Sates.
  • Skorupinska-Tudek K; Department of Lipid Biochemistry, Institute of Biochemistry and Biophysics, Polish Academy of Sciences, Pawinskiego 5a, 02-106 Warszawa, Poland.
  • Swiezewska E; Department of Lipid Biochemistry, Institute of Biochemistry and Biophysics, Polish Academy of Sciences, Pawinskiego 5a, 02-106 Warszawa, Poland.
  • Franzblau SG; Institute for Tuberculosis Research, College of Pharmacy, University of Illinois at Chicago, 833 S. Wood Street, Chicago, IL 60612, United States.
  • Kurosu M; Department of Pharmaceutical Sciences, College of Pharmacy, University of Tennessee Health Science Center, 881 Madison Avenue, Memphis, TN 38163-0001, United States. Electronic address: mkurosu@uthsc.edu.
Anal Biochem ; 512: 78-90, 2016 11 01.
Article en En | MEDLINE | ID: mdl-27530653

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Proteínas Bacterianas / Transferasas (Grupos de Otros Fosfatos Sustitutos) / Inhibidores Enzimáticos / Mycobacterium tuberculosis / Antituberculosos Tipo de estudio: Diagnostic_studies Idioma: En Revista: Anal Biochem Año: 2016 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Proteínas Bacterianas / Transferasas (Grupos de Otros Fosfatos Sustitutos) / Inhibidores Enzimáticos / Mycobacterium tuberculosis / Antituberculosos Tipo de estudio: Diagnostic_studies Idioma: En Revista: Anal Biochem Año: 2016 Tipo del documento: Article País de afiliación: Estados Unidos