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Inhibitor mechanisms in the S1 binding site of the dopamine transporter defined by multi-site molecular tethering of photoactive cocaine analogs.
Krout, Danielle; Pramod, Akula Bala; Dahal, Rejwi Acharya; Tomlinson, Michael J; Sharma, Babita; Foster, James D; Zou, Mu-Fa; Boatang, Comfort; Newman, Amy Hauck; Lever, John R; Vaughan, Roxanne A; Henry, L Keith.
Afiliación
  • Krout D; Department of Biomedical Sciences, University of North Dakota School of Medicine and Health Sciences, 1301 North Columbia Road, Grand Forks, ND 58202, USA.
  • Pramod AB; Department of Biomedical Sciences, University of North Dakota School of Medicine and Health Sciences, 1301 North Columbia Road, Grand Forks, ND 58202, USA.
  • Dahal RA; Department of Biomedical Sciences, University of North Dakota School of Medicine and Health Sciences, 1301 North Columbia Road, Grand Forks, ND 58202, USA.
  • Tomlinson MJ; Department of Biomedical Sciences, University of North Dakota School of Medicine and Health Sciences, 1301 North Columbia Road, Grand Forks, ND 58202, USA.
  • Sharma B; Department of Biomedical Sciences, University of North Dakota School of Medicine and Health Sciences, 1301 North Columbia Road, Grand Forks, ND 58202, USA.
  • Foster JD; Department of Biomedical Sciences, University of North Dakota School of Medicine and Health Sciences, 1301 North Columbia Road, Grand Forks, ND 58202, USA.
  • Zou MF; Medicinal Chemistry Section, National Institute on Drug Abuse - Intramural Research Program, Baltimore, MD 21224, USA.
  • Boatang C; Medicinal Chemistry Section, National Institute on Drug Abuse - Intramural Research Program, Baltimore, MD 21224, USA.
  • Newman AH; Medicinal Chemistry Section, National Institute on Drug Abuse - Intramural Research Program, Baltimore, MD 21224, USA.
  • Lever JR; Research Service, Harry S. Truman Memorial Veterans' Hospital, Columbia, MO, 65201, USA; Department of Radiology and Radiopharmaceutical Sciences Institute, University of Missouri, Columbia, MO 65211, USA.
  • Vaughan RA; Department of Biomedical Sciences, University of North Dakota School of Medicine and Health Sciences, 1301 North Columbia Road, Grand Forks, ND 58202, USA. Electronic address: roxanne.vaughan@med.und.edu.
  • Henry LK; Department of Biomedical Sciences, University of North Dakota School of Medicine and Health Sciences, 1301 North Columbia Road, Grand Forks, ND 58202, USA. Electronic address: keith.henry@med.und.edu.
Biochem Pharmacol ; 142: 204-215, 2017 10 15.
Article en En | MEDLINE | ID: mdl-28734777

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Tropanos / Cocaína / Trastornos Relacionados con Sustancias / Proteínas de Transporte de Dopamina a través de la Membrana Plasmática Tipo de estudio: Prognostic_studies Idioma: En Revista: Biochem Pharmacol Año: 2017 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Tropanos / Cocaína / Trastornos Relacionados con Sustancias / Proteínas de Transporte de Dopamina a través de la Membrana Plasmática Tipo de estudio: Prognostic_studies Idioma: En Revista: Biochem Pharmacol Año: 2017 Tipo del documento: Article País de afiliación: Estados Unidos