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Identification of Bichalcones as Sirtuin Inhibitors by Virtual Screening and In Vitro Testing.
Karaman, Berin; Alhalabi, Zayan; Swyter, Sören; Mihigo, Shetonde O; Andrae-Marobela, Kerstin; Jung, Manfred; Sippl, Wolfgang; Ntie-Kang, Fidele.
Afiliación
  • Karaman B; Department of Pharmaceutical Chemistry, Martin-Luther University of Halle-Wittenberg, Wolfgang-Langenbeck-Str. 4, 06120 Halle (Saale), Germany. karaman.berin@gmail.com.
  • Alhalabi Z; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Biruni University, Istanbul 34010, Turkey. karaman.berin@gmail.com.
  • Swyter S; Department of Pharmaceutical Chemistry, Martin-Luther University of Halle-Wittenberg, Wolfgang-Langenbeck-Str. 4, 06120 Halle (Saale), Germany. zayan82at@hotmail.com.
  • Mihigo SO; Institute of Pharmaceutical Sciences, Albert-Ludwigs-University of Freiburg, Albertstr. 25, 79104 Freiburg im Breisgau, Germany. soeren.swyter@pharmazie.uni-freiburg.de.
  • Andrae-Marobela K; Department of Chemistry, University of Kinshasa, Kinshasa P.O. Box 190 XI, Congo. smihigo@yahoo.com.
  • Jung M; Department of Biological Sciences, Faculty of Science, University of Botswana, Block 235, Private Bag, Gaborone 0022, Botswana. k_marobela@yahoo.com.
  • Sippl W; Institute of Pharmaceutical Sciences, Albert-Ludwigs-University of Freiburg, Albertstr. 25, 79104 Freiburg im Breisgau, Germany. manfred.jung@pharmazie.uni-freiburg.de.
  • Ntie-Kang F; Department of Pharmaceutical Chemistry, Martin-Luther University of Halle-Wittenberg, Wolfgang-Langenbeck-Str. 4, 06120 Halle (Saale), Germany. wolfgang.sippl@pharmazie.uni-halle.de.
Molecules ; 23(2)2018 Feb 14.
Article en En | MEDLINE | ID: mdl-29443909

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Chalconas / Sirtuina 1 / Inhibidores de Histona Desacetilasas Tipo de estudio: Diagnostic_studies / Screening_studies Idioma: En Revista: Molecules Año: 2018 Tipo del documento: Article País de afiliación: Alemania

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Chalconas / Sirtuina 1 / Inhibidores de Histona Desacetilasas Tipo de estudio: Diagnostic_studies / Screening_studies Idioma: En Revista: Molecules Año: 2018 Tipo del documento: Article País de afiliación: Alemania