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Optimization of 4-arylthiophene-3-carboxylic acid derivatives as inhibitors of ANO1: Lead optimization studies toward their analgesic efficacy for inflammatory pain.
Wang, Yuxi; Hu, Xiaoyue; Huang, Han; Jin, Zefang; Gao, Jian; Guo, Yi; Zhong, Yi; Li, Zhongtang; Zong, Xiaolin; Wang, Kewei; Zhang, Liangren; Liu, Zhenming.
Afiliación
  • Wang Y; State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing, 100191, China.
  • Hu X; State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing, 100191, China.
  • Huang H; State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing, 100191, China.
  • Jin Z; State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing, 100191, China.
  • Gao J; State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing, 100191, China.
  • Guo Y; State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing, 100191, China.
  • Zhong Y; State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing, 100191, China.
  • Li Z; State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing, 100191, China.
  • Zong X; State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing, 100191, China.
  • Wang K; Department of Pharmacology, School of Pharmacy, Qingdao University, Qingdao, 266021, China.
  • Zhang L; State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing, 100191, China. Electronic address: liangren@bjmu.edu.cn.
  • Liu Z; State Key Laboratory of Natural and Biomimetic Drugs, School of Pharmaceutical Sciences, Peking University, Beijing, 100191, China. Electronic address: zmliu@bjmu.edu.cn.
Eur J Med Chem ; 237: 114413, 2022 Jul 05.
Article en En | MEDLINE | ID: mdl-35512566

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Dolor / Analgésicos Idioma: En Revista: Eur J Med Chem Año: 2022 Tipo del documento: Article País de afiliación: China

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Dolor / Analgésicos Idioma: En Revista: Eur J Med Chem Año: 2022 Tipo del documento: Article País de afiliación: China