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Identification of novel PTP1B inhibitors by pharmacophore based virtual screening, scaffold hopping and docking.
Balaramnavar, Vishal M; Srivastava, Rohit; Rahuja, Neha; Gupta, Swati; Rawat, Arun K; Varshney, Salil; Chandasana, Hardik; Chhonker, Yashpal S; Doharey, Pawan Kumar; Kumar, Santosh; Gautam, Sudeep; Srivastava, Swayam Prakash; Bhatta, Rabi Sankar; Saxena, Jitendra Kumar; Gaikwad, Anil Nilkanth; Srivastava, Arvind K; Saxena, Anil K.
Afiliação
  • Balaramnavar VM; Division of Medicinal and Process Chemistry, CSIR-Central Drug Research Institute, Jankipuram Extension, Lucknow 226021, UP, India.
  • Srivastava R; Division of Biochemistry, Central Drug Research Institute, CSIR, Jankipuram Extension, Lucknow 226021, UP, India.
  • Rahuja N; Division of Biochemistry, Central Drug Research Institute, CSIR, Jankipuram Extension, Lucknow 226021, UP, India.
  • Gupta S; Division of Medicinal and Process Chemistry, CSIR-Central Drug Research Institute, Jankipuram Extension, Lucknow 226021, UP, India.
  • Rawat AK; Division of Biochemistry, Central Drug Research Institute, CSIR, Jankipuram Extension, Lucknow 226021, UP, India.
  • Varshney S; Division of Pharmacology, CSIR-Central Drug Research Institute, Jankipuram Extension, Lucknow 226021, UP, India.
  • Chandasana H; Pharmacokinetics and Metabolism Division, CSIR-Central Drug Research Institute, Jankipuram Extension, Lucknow 226021, UP, India.
  • Chhonker YS; Pharmacokinetics and Metabolism Division, CSIR-Central Drug Research Institute, Jankipuram Extension, Lucknow 226021, UP, India.
  • Doharey PK; Division of Biochemistry, Central Drug Research Institute, CSIR, Jankipuram Extension, Lucknow 226021, UP, India.
  • Kumar S; Division of Medicinal and Process Chemistry, CSIR-Central Drug Research Institute, Jankipuram Extension, Lucknow 226021, UP, India.
  • Gautam S; Division of Biochemistry, Central Drug Research Institute, CSIR, Jankipuram Extension, Lucknow 226021, UP, India.
  • Srivastava SP; Division of Biochemistry, Central Drug Research Institute, CSIR, Jankipuram Extension, Lucknow 226021, UP, India.
  • Bhatta RS; Pharmacokinetics and Metabolism Division, CSIR-Central Drug Research Institute, Jankipuram Extension, Lucknow 226021, UP, India.
  • Saxena JK; Division of Biochemistry, Central Drug Research Institute, CSIR, Jankipuram Extension, Lucknow 226021, UP, India.
  • Gaikwad AN; Division of Pharmacology, CSIR-Central Drug Research Institute, Jankipuram Extension, Lucknow 226021, UP, India.
  • Srivastava AK; Division of Biochemistry, Central Drug Research Institute, CSIR, Jankipuram Extension, Lucknow 226021, UP, India.
  • Saxena AK; Division of Medicinal and Process Chemistry, CSIR-Central Drug Research Institute, Jankipuram Extension, Lucknow 226021, UP, India. Electronic address: anilsak@gmail.com.
Eur J Med Chem ; 87: 578-94, 2014 Nov 24.
Article em En | MEDLINE | ID: mdl-25299681

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores Enzimáticos / Proteína Tirosina Fosfatase não Receptora Tipo 1 Tipo de estudo: Diagnostic_studies / Screening_studies Idioma: En Revista: Eur J Med Chem Ano de publicação: 2014 Tipo de documento: Article País de afiliação: Índia

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores Enzimáticos / Proteína Tirosina Fosfatase não Receptora Tipo 1 Tipo de estudo: Diagnostic_studies / Screening_studies Idioma: En Revista: Eur J Med Chem Ano de publicação: 2014 Tipo de documento: Article País de afiliação: Índia