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Glucuronidation of bavachinin by human tissues and expressed UGT enzymes: Identification of UGT1A1 and UGT1A8 as the major contributing enzymes.
Lv, Xia; Hou, Jie; Xia, Yang-Liu; Ning, Jing; He, Gui-Yuan; Wang, Ping; Ge, Guang-Bo; Xiu, Zhi-Long; Yang, Ling.
Afiliação
  • Lv X; Department of Bioscience and Biotechnology, Dalian University of Technology, Dalian, China; Laboratory of Pharmaceutical Resource Discovery, Dalian Institute of Chemical Physics, Chinese Academy of Sciences, Dalian, China.
  • Hou J; Dalian Medical University, Dalian, China.
  • Xia YL; Laboratory of Pharmaceutical Resource Discovery, Dalian Institute of Chemical Physics, Chinese Academy of Sciences, Dalian, China.
  • Ning J; Laboratory of Pharmaceutical Resource Discovery, Dalian Institute of Chemical Physics, Chinese Academy of Sciences, Dalian, China; Dalian Medical University, Dalian, China.
  • He GY; Laboratory of Pharmaceutical Resource Discovery, Dalian Institute of Chemical Physics, Chinese Academy of Sciences, Dalian, China.
  • Wang P; Laboratory of Pharmaceutical Resource Discovery, Dalian Institute of Chemical Physics, Chinese Academy of Sciences, Dalian, China.
  • Ge GB; Laboratory of Pharmaceutical Resource Discovery, Dalian Institute of Chemical Physics, Chinese Academy of Sciences, Dalian, China. Electronic address: geguangbo@dicp.ac.cn.
  • Xiu ZL; Department of Bioscience and Biotechnology, Dalian University of Technology, Dalian, China.
  • Yang L; Laboratory of Pharmaceutical Resource Discovery, Dalian Institute of Chemical Physics, Chinese Academy of Sciences, Dalian, China. Electronic address: ylingdicp@gmail.com.
Drug Metab Pharmacokinet ; 30(5): 358-65, 2015 Oct.
Article em En | MEDLINE | ID: mdl-26320626

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Flavonoides / Glucuronosiltransferase Tipo de estudo: Diagnostic_studies / Prognostic_studies Idioma: En Revista: Drug Metab Pharmacokinet Ano de publicação: 2015 Tipo de documento: Article País de afiliação: China

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Flavonoides / Glucuronosiltransferase Tipo de estudo: Diagnostic_studies / Prognostic_studies Idioma: En Revista: Drug Metab Pharmacokinet Ano de publicação: 2015 Tipo de documento: Article País de afiliação: China