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Pharmacological Evaluation of Novel Bioisosteres of an Adamantanyl Benzamide P2X7 Receptor Antagonist.
Wilkinson, Shane M; Barron, Melissa L; O'Brien-Brown, James; Janssen, Bieneke; Stokes, Leanne; Werry, Eryn L; Chishty, Mansoor; Skarratt, Kristen K; Ong, Jennifer A; Hibbs, David E; Vugts, Danielle J; Fuller, Stephen; Windhorst, Albert D; Kassiou, Michael.
Afiliação
  • Janssen B; Department of Radiology & Nuclear Medicine, VU University Medical Center , De Boelelaan 1117, 1081 HV Amsterdam, The Netherlands.
  • Stokes L; School of Pharmacy, University of East Anglia , Norwich NR4 7TJ, U.K.
  • Chishty M; Pharmidex , 14 Hanover St., Mayfair, London W1S 1YH, U.K.
  • Vugts DJ; Department of Radiology & Nuclear Medicine, VU University Medical Center , De Boelelaan 1117, 1081 HV Amsterdam, The Netherlands.
  • Windhorst AD; Department of Radiology & Nuclear Medicine, VU University Medical Center , De Boelelaan 1117, 1081 HV Amsterdam, The Netherlands.
ACS Chem Neurosci ; 8(11): 2374-2380, 2017 11 15.
Article em En | MEDLINE | ID: mdl-28841278

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Benzamidas / Adamantano / Receptores Purinérgicos P2X7 / Antagonistas do Receptor Purinérgico P2X Idioma: En Revista: ACS Chem Neurosci Ano de publicação: 2017 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Benzamidas / Adamantano / Receptores Purinérgicos P2X7 / Antagonistas do Receptor Purinérgico P2X Idioma: En Revista: ACS Chem Neurosci Ano de publicação: 2017 Tipo de documento: Article