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Identification of Cyanamide-Based Janus Kinase 3 (JAK3) Covalent Inhibitors.
Casimiro-Garcia, Agustin; Trujillo, John I; Vajdos, Felix; Juba, Brian; Banker, Mary Ellen; Aulabaugh, Ann; Balbo, Paul; Bauman, Jonathan; Chrencik, Jill; Coe, Jotham W; Czerwinski, Robert; Dowty, Martin; Knafels, John D; Kwon, Soojin; Leung, Louis; Liang, Sidney; Robinson, Ralph P; Telliez, Jean-Baptiste; Unwalla, Ray; Yang, Xin; Thorarensen, Atli.
Afiliação
  • Trujillo JI; Medicine Design , Pfizer Inc. , 445 Eastern Point Road , Groton , Connecticut 06340 , United States.
  • Vajdos F; Medicine Design , Pfizer Inc. , 445 Eastern Point Road , Groton , Connecticut 06340 , United States.
  • Banker ME; Medicine Design , Pfizer Inc. , 445 Eastern Point Road , Groton , Connecticut 06340 , United States.
  • Aulabaugh A; Medicine Design , Pfizer Inc. , 445 Eastern Point Road , Groton , Connecticut 06340 , United States.
  • Bauman J; Medicine Design , Pfizer Inc. , 445 Eastern Point Road , Groton , Connecticut 06340 , United States.
  • Chrencik J; Medicine Design , Pfizer Inc. , 445 Eastern Point Road , Groton , Connecticut 06340 , United States.
  • Coe JW; Medicine Design , Pfizer Inc. , 445 Eastern Point Road , Groton , Connecticut 06340 , United States.
  • Dowty M; Medicine Design , Pfizer Inc. , 1 Burtt Road , Andover , Massachusetts 01810 , United States.
  • Knafels JD; Medicine Design , Pfizer Inc. , 445 Eastern Point Road , Groton , Connecticut 06340 , United States.
  • Kwon S; Medicine Design , Pfizer Inc. , 445 Eastern Point Road , Groton , Connecticut 06340 , United States.
  • Leung L; Medicine Design , Pfizer Inc. , 445 Eastern Point Road , Groton , Connecticut 06340 , United States.
  • Liang S; Medicine Design , Pfizer Inc. , 445 Eastern Point Road , Groton , Connecticut 06340 , United States.
  • Robinson RP; Medicine Design , Pfizer Inc. , 445 Eastern Point Road , Groton , Connecticut 06340 , United States.
  • Yang X; Medicine Design , Pfizer Inc. , 445 Eastern Point Road , Groton , Connecticut 06340 , United States.
J Med Chem ; 61(23): 10665-10699, 2018 12 13.
Article em En | MEDLINE | ID: mdl-30423248

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Cianamida / Inibidores de Proteínas Quinases / Janus Quinase 3 Tipo de estudo: Diagnostic_studies Idioma: En Revista: J Med Chem Ano de publicação: 2018 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Cianamida / Inibidores de Proteínas Quinases / Janus Quinase 3 Tipo de estudo: Diagnostic_studies Idioma: En Revista: J Med Chem Ano de publicação: 2018 Tipo de documento: Article