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Static Model-Based Assessment of OATP1B1-Mediated Drug Interactions with Preincubation-Dependent Inhibitors Based on Inactivation and Recovery Kinetics.
Taguchi, Takayuki; Masuo, Yusuke; Futatsugi, Azusa; Kato, Yukio.
Afiliação
  • Taguchi T; Pharmacokinetics and Safety Department, Drug Research Center, Kaken Pharmaceutical Co., Ltd., Kyoto, Japan (T.T.) and Faculty of Pharmacy, Institute of Medical, Pharmaceutical and Health Sciences, Kanazawa University, Kanazawa, Japan (T.T., Y.M., A.F., Y.K.).
  • Masuo Y; Pharmacokinetics and Safety Department, Drug Research Center, Kaken Pharmaceutical Co., Ltd., Kyoto, Japan (T.T.) and Faculty of Pharmacy, Institute of Medical, Pharmaceutical and Health Sciences, Kanazawa University, Kanazawa, Japan (T.T., Y.M., A.F., Y.K.).
  • Futatsugi A; Pharmacokinetics and Safety Department, Drug Research Center, Kaken Pharmaceutical Co., Ltd., Kyoto, Japan (T.T.) and Faculty of Pharmacy, Institute of Medical, Pharmaceutical and Health Sciences, Kanazawa University, Kanazawa, Japan (T.T., Y.M., A.F., Y.K.).
  • Kato Y; Pharmacokinetics and Safety Department, Drug Research Center, Kaken Pharmaceutical Co., Ltd., Kyoto, Japan (T.T.) and Faculty of Pharmacy, Institute of Medical, Pharmaceutical and Health Sciences, Kanazawa University, Kanazawa, Japan (T.T., Y.M., A.F., Y.K.) ykato@p.kanazawa-u.ac.jp.
Drug Metab Dispos ; 48(9): 750-758, 2020 09.
Article em En | MEDLINE | ID: mdl-32616544

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Transportador 1 de Ânion Orgânico Específico do Fígado / Interações Medicamentosas / Eliminação Hepatobiliar / Modelos Biológicos Tipo de estudo: Prognostic_studies Idioma: En Revista: Drug Metab Dispos Ano de publicação: 2020 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Transportador 1 de Ânion Orgânico Específico do Fígado / Interações Medicamentosas / Eliminação Hepatobiliar / Modelos Biológicos Tipo de estudo: Prognostic_studies Idioma: En Revista: Drug Metab Dispos Ano de publicação: 2020 Tipo de documento: Article