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Ligand-Induced Conformational Change of Insulin-Regulated Aminopeptidase: Insights on Catalytic Mechanism and Active Site Plasticity.
Mpakali, Anastasia; Saridakis, Emmanuel; Harlos, Karl; Zhao, Yuguang; Kokkala, Paraskevi; Georgiadis, Dimitris; Giastas, Petros; Papakyriakou, Athanasios; Stratikos, Efstratios.
Afiliación
  • Mpakali A; National Center for Scientific Research Demokritos, Agia Paraskevi , Athens 15310, Greece.
  • Saridakis E; National Center for Scientific Research Demokritos, Agia Paraskevi , Athens 15310, Greece.
  • Harlos K; Division of Structural Biology, Wellcome Trust Centre for Human Genetics, Oxford University , Oxford OX3 7BN, United Kingdom.
  • Zhao Y; Division of Structural Biology, Wellcome Trust Centre for Human Genetics, Oxford University , Oxford OX3 7BN, United Kingdom.
  • Kokkala P; Department of Chemistry, University of Athens , Athens 15771, Greece.
  • Georgiadis D; Department of Chemistry, University of Athens , Athens 15771, Greece.
  • Giastas P; National Center for Scientific Research Demokritos, Agia Paraskevi , Athens 15310, Greece.
  • Papakyriakou A; National Center for Scientific Research Demokritos, Agia Paraskevi , Athens 15310, Greece.
  • Stratikos E; National Center for Scientific Research Demokritos, Agia Paraskevi , Athens 15310, Greece.
J Med Chem ; 60(7): 2963-2972, 2017 04 13.
Article en En | MEDLINE | ID: mdl-28328206

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Cistinil Aminopeptidasa / Conformación Proteica / Inhibidores Enzimáticos Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2017 Tipo del documento: Article

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Cistinil Aminopeptidasa / Conformación Proteica / Inhibidores Enzimáticos Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2017 Tipo del documento: Article