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Design, synthesis, and biological evaluation of aryl N-methoxyamide derivatives as GPR119 agonists.
Jang, Yoon Kyung; Lee, Kyu Myung; Jung, Kwan-Young; Kang, Seung Kyu; Pagire, Suvarna H; Lee, Jun Mi; Pagire, Haushabhau S; Kim, Kwang Rok; Bae, Myung Ae; Lee, Hohjai; Rhee, Sang Dal; Ahn, Jin Hee.
Afiliación
  • Jang YK; Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 305-600, Republic of Korea.
  • Lee KM; Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 305-600, Republic of Korea.
  • Jung KY; Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 305-600, Republic of Korea.
  • Kang SK; Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 305-600, Republic of Korea.
  • Pagire SH; Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 305-600, Republic of Korea.
  • Lee JM; Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 305-600, Republic of Korea.
  • Pagire HS; Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 305-600, Republic of Korea.
  • Kim KR; Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 305-600, Republic of Korea.
  • Bae MA; Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 305-600, Republic of Korea.
  • Lee H; Department of Chemistry, Gwangju Institute of Science and Technology, Gwangju 61005, Republic of Korea.
  • Rhee SD; Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 305-600, Republic of Korea.
  • Ahn JH; Drug Discovery Division, Korea Research Institute of Chemical Technology, Daejeon 305-600, Republic of Korea; Department of Chemistry, Gwangju Institute of Science and Technology, Gwangju 61005, Republic of Korea. Electronic address: jhahn@gist.ac.kr.
Bioorg Med Chem Lett ; 27(16): 3909-3914, 2017 08 15.
Article en En | MEDLINE | ID: mdl-28666737

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Diseño de Fármacos / Receptores Acoplados a Proteínas G / Amidas Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2017 Tipo del documento: Article

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Diseño de Fármacos / Receptores Acoplados a Proteínas G / Amidas Idioma: En Revista: Bioorg Med Chem Lett Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2017 Tipo del documento: Article