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Two key cathepsins, TgCPB and TgCPL, are targeted by the vinyl sulfone inhibitor K11777 in in vitro and in vivo models of toxoplasmosis.
Chaparro, Juan D; Cheng, Timmy; Tran, Uyen Phuong; Andrade, Rosa M; Brenner, Sara B T; Hwang, Grace; Cohn, Shara; Hirata, Ken; McKerrow, James H; Reed, Sharon L.
Afiliación
  • Chaparro JD; Department of Pediatrics, Division of Infectious Diseases, Rady Children's Hospital, University of California, San Diego, School of Medicine, La Jolla, California, United States of America.
  • Cheng T; Department of Pathology, University of California, San Diego School of Medicine, La Jolla, California, United States of America.
  • Tran UP; Department of Pathology, University of California, San Diego School of Medicine, La Jolla, California, United States of America.
  • Andrade RM; Department of Medicine, Division of Infectious Diseases, University of California, Irvine School of Medicine, Irvine, California, United States of America.
  • Brenner SBT; Department of Pathology, University of California, San Diego School of Medicine, La Jolla, California, United States of America.
  • Hwang G; Department of Pathology, University of California, San Diego School of Medicine, La Jolla, California, United States of America.
  • Cohn S; Department of Pathology, University of California, San Diego School of Medicine, La Jolla, California, United States of America.
  • Hirata K; Department of Pathology, University of California, San Diego School of Medicine, La Jolla, California, United States of America.
  • McKerrow JH; Department of Pharmacy, Skaggs School of Pharmacy and Pharmaceutical Science, University of California, San Diego, La Jolla, California, United States of America.
  • Reed SL; Department of Pathology, University of California, San Diego School of Medicine, La Jolla, California, United States of America.
PLoS One ; 13(3): e0193982, 2018.
Article en En | MEDLINE | ID: mdl-29565998

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Sulfonas / Compuestos de Vinilo / Catepsinas / Proteínas Protozoarias / Toxoplasmosis / Dipéptidos Idioma: En Revista: PLoS One Asunto de la revista: CIENCIA / MEDICINA Año: 2018 Tipo del documento: Article

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Sulfonas / Compuestos de Vinilo / Catepsinas / Proteínas Protozoarias / Toxoplasmosis / Dipéptidos Idioma: En Revista: PLoS One Asunto de la revista: CIENCIA / MEDICINA Año: 2018 Tipo del documento: Article