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Discovery of Tyrosine Kinase 2 (TYK2) Inhibitor (PF-06826647) for the Treatment of Autoimmune Diseases.
Gerstenberger, Brian S; Ambler, Catherine; Arnold, Eric P; Banker, Mary-Ellen; Brown, Matthew F; Clark, James D; Dermenci, Alpay; Dowty, Martin E; Fensome, Andrew; Fish, Susan; Hayward, Matthew M; Hegen, Martin; Hollingshead, Brett D; Knafels, John D; Lin, David W; Lin, Tsung H; Owen, Dafydd R; Saiah, Eddine; Sharma, Raman; Vajdos, Felix F; Xing, Li; Yang, Xiaojing; Yang, Xin; Wright, Stephen W.
Afiliación
  • Gerstenberger BS; Pfizer Inc., Cambridge, Massachusetts 02139, United States.
  • Ambler C; Pfizer Inc., Groton, Connecticut 06340, United States.
  • Arnold EP; Pfizer Inc., Groton, Connecticut 06340, United States.
  • Banker ME; Pfizer Inc., Groton, Connecticut 06340, United States.
  • Brown MF; Pfizer Inc., Groton, Connecticut 06340, United States.
  • Clark JD; Pfizer Inc., Cambridge, Massachusetts 02139, United States.
  • Dermenci A; Pfizer Inc., Groton, Connecticut 06340, United States.
  • Dowty ME; Pfizer Inc., Cambridge, Massachusetts 02139, United States.
  • Fensome A; Pfizer Inc., Cambridge, Massachusetts 02139, United States.
  • Fish S; Pfizer Inc., Cambridge, Massachusetts 02139, United States.
  • Hayward MM; Pfizer Inc., Groton, Connecticut 06340, United States.
  • Hegen M; Pfizer Inc., Cambridge, Massachusetts 02139, United States.
  • Hollingshead BD; Pfizer Inc., Cambridge, Massachusetts 02139, United States.
  • Knafels JD; Pfizer Inc., Groton, Connecticut 06340, United States.
  • Lin DW; Pfizer Inc., Groton, Connecticut 06340, United States.
  • Lin TH; Pfizer Inc., Cambridge, Massachusetts 02139, United States.
  • Owen DR; Pfizer Inc., Cambridge, Massachusetts 02139, United States.
  • Saiah E; Pfizer Inc., Cambridge, Massachusetts 02139, United States.
  • Sharma R; Pfizer Inc., Groton, Connecticut 06340, United States.
  • Vajdos FF; Pfizer Inc., Groton, Connecticut 06340, United States.
  • Xing L; Pfizer Inc., Cambridge, Massachusetts 02139, United States.
  • Yang X; Pfizer Inc., Groton, Connecticut 06340, United States.
  • Yang X; Pfizer Inc., Groton, Connecticut 06340, United States.
  • Wright SW; Pfizer Inc., Groton, Connecticut 06340, United States.
J Med Chem ; 63(22): 13561-13577, 2020 11 25.
Article en En | MEDLINE | ID: mdl-32787094

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Enfermedades Autoinmunes / Inhibidores de Proteínas Quinasas / TYK2 Quinasa / Descubrimiento de Drogas Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2020 Tipo del documento: Article

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Enfermedades Autoinmunes / Inhibidores de Proteínas Quinasas / TYK2 Quinasa / Descubrimiento de Drogas Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2020 Tipo del documento: Article