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Mechanism-Based Inactivation of Cytochrome P450 3A4 and 3A5 by the Fibroblast Growth Factor Receptor Inhibitor Erdafitinib.
Tang, Lloyd Wei Tat; Teng, Jian Wei; Koh, Siew Kwan; Zhou, Lei; Go, Mei Lin; Chan, Eric Chun Yong.
Afiliación
  • Tang LWT; Department of Pharmacy, Faculty of Science, National University of Singapore, 169856 Singapore.
  • Teng JW; Department of Pharmacy, Faculty of Science, National University of Singapore, 169856 Singapore.
  • Koh SK; Singapore Eye Research Institute (SERI), Singapore.
  • Zhou L; Singapore Eye Research Institute (SERI), Singapore.
  • Go ML; Department of Ophthalmology, Yong Loo Lin School of Medicine, National University of Singapore, 117597 Singapore.
  • Chan ECY; Ophthalmology and Visual Sciences Academia Clinical Program, Duke-National University of Singapore Medical School, 169857 Singapore.
Chem Res Toxicol ; 34(7): 1800-1813, 2021 07 19.
Article en En | MEDLINE | ID: mdl-34189909

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Pirazoles / Quinoxalinas / Receptores de Factores de Crecimiento de Fibroblastos / Inhibidores del Citocromo P-450 CYP3A Idioma: En Revista: Chem Res Toxicol Asunto de la revista: TOXICOLOGIA Año: 2021 Tipo del documento: Article

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Pirazoles / Quinoxalinas / Receptores de Factores de Crecimiento de Fibroblastos / Inhibidores del Citocromo P-450 CYP3A Idioma: En Revista: Chem Res Toxicol Asunto de la revista: TOXICOLOGIA Año: 2021 Tipo del documento: Article