Comparison of anti-SARS-CoV-2 activity and intracellular metabolism of remdesivir and its parent nucleoside.
Curr Res Pharmacol Drug Discov
; 2: 100045, 2021.
Article
en En
| MEDLINE
| ID: mdl-34870151
ACE2, angiotensin-converting enzyme 2; Anti-SARS-CoV-2; Antiviral agents; CES1, carboxylesterase 1; COVID-19; COVID-19, coronavirus disease 2019; CatA, cathepsin A; Coronavirus; DP, diphosphate; GS-441524; HAE, human airway epithelial; HCoV-OC43; HINT1, histidine triad nucleotide-binding protein 1; MP, monophosphate; NTP, nucleoside triphosphate; Pharmacology; Remdesivir; SARS-CoV-2, severe acute respiratory syndrome coronavirus 2; TP, triphosphate; WHO, World Health Organization; icSARS-CoV-2-mNG, SARS-CoV-2 infectious clone virus containing mNeonGreen reporter
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Curr Res Pharmacol Drug Discov
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2021
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