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Discovery of a New Drug-like Series of OGT Inhibitors by Virtual Screening.
Loi, Elena M; Tomasic, Tihomir; Balsollier, Cyril; van Eekelen, Kevin; Weiss, Matjaz; Gobec, Martina; Alteen, Matthew G; Vocadlo, David J; Pieters, Roland J; Anderluh, Marko.
Afiliación
  • Loi EM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Ljubljana, 1000 Ljubljana, Slovenia.
  • Tomasic T; Department of Chemical Biology & Drug Discovery, Utrecht Institute for Pharmaceutical Sciences, Utrecht University, 3584 CG Utrecht, The Netherlands.
  • Balsollier C; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Ljubljana, 1000 Ljubljana, Slovenia.
  • van Eekelen K; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Ljubljana, 1000 Ljubljana, Slovenia.
  • Weiss M; Department of Chemical Biology & Drug Discovery, Utrecht Institute for Pharmaceutical Sciences, Utrecht University, 3584 CG Utrecht, The Netherlands.
  • Gobec M; Department of Chemical Biology & Drug Discovery, Utrecht Institute for Pharmaceutical Sciences, Utrecht University, 3584 CG Utrecht, The Netherlands.
  • Alteen MG; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Ljubljana, 1000 Ljubljana, Slovenia.
  • Vocadlo DJ; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Ljubljana, 1000 Ljubljana, Slovenia.
  • Pieters RJ; Department of Chemistry, Simon Fraser University, Burnaby, BC V5A 1S6, Canada.
  • Anderluh M; Department of Chemistry, Simon Fraser University, Burnaby, BC V5A 1S6, Canada.
Molecules ; 27(6)2022 Mar 19.
Article en En | MEDLINE | ID: mdl-35335358

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Procesamiento Proteico-Postraduccional / N-Acetilglucosaminiltransferasas Tipo de estudio: Diagnostic_studies / Screening_studies Idioma: En Revista: Molecules Asunto de la revista: BIOLOGIA Año: 2022 Tipo del documento: Article

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Procesamiento Proteico-Postraduccional / N-Acetilglucosaminiltransferasas Tipo de estudio: Diagnostic_studies / Screening_studies Idioma: En Revista: Molecules Asunto de la revista: BIOLOGIA Año: 2022 Tipo del documento: Article