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5-Alkoxy-1-aryl-3-polyfluoroalkylpyrazoles with Antinociceptive Activity: Partial Agonists of TRPV1 Ion Channels.
Khudina, Olga G; Burgart, Yanina V; Malkova, Natalia A; Shchegolkov, Evgeny V; Krasnykh, Olga P; Triandafilova, Galina A; Malysheva, Ksenia O; Solodnikov, Sergey Yu; Dubodel, Elisaveta S; Korolkova, Yuliya V; Kozlov, Sergey A; Borisevich, Sophia S; Mozhaitsev, Evgenii S; Saloutin, Victor I.
Afiliación
  • Khudina OG; Ural Branch of the Russian Academy of Sciences, Postovsky Institute of Organic Synthesis, S. Kovalevskoi St., 22, Ekaterinburg, 620108, Russia.
  • Burgart YV; Ural Branch of the Russian Academy of Sciences, Postovsky Institute of Organic Synthesis, S. Kovalevskoi St., 22, Ekaterinburg, 620108, Russia.
  • Malkova NA; Ural Branch of the Russian Academy of Sciences, Postovsky Institute of Organic Synthesis, S. Kovalevskoi St., 22, Ekaterinburg, 620108, Russia.
  • Shchegolkov EV; Ural Branch of the Russian Academy of Sciences, Postovsky Institute of Organic Synthesis, S. Kovalevskoi St., 22, Ekaterinburg, 620108, Russia.
  • Krasnykh OP; Scientific and Educational Center for Applied Chemical-Biological Research, Perm National Research Polytechnic University, Komsomolsky Av., 29, Perm, 614990, Russia.
  • Triandafilova GA; Scientific and Educational Center for Applied Chemical-Biological Research, Perm National Research Polytechnic University, Komsomolsky Av., 29, Perm, 614990, Russia.
  • Malysheva KO; Scientific and Educational Center for Applied Chemical-Biological Research, Perm National Research Polytechnic University, Komsomolsky Av., 29, Perm, 614990, Russia.
  • Solodnikov SY; Scientific and Educational Center for Applied Chemical-Biological Research, Perm National Research Polytechnic University, Komsomolsky Av., 29, Perm, 614990, Russia.
  • Dubodel ES; The Russian Academy of Sciences, Shemyakin-Ovchinnikov Institute of Bioorganic Chemistry, Miklukho-Maklaya St., 16/10, Moscow, 117997, Russia.
  • Korolkova YV; The Russian Academy of Sciences, Shemyakin-Ovchinnikov Institute of Bioorganic Chemistry, Miklukho-Maklaya St., 16/10, Moscow, 117997, Russia.
  • Kozlov SA; The Russian Academy of Sciences, Shemyakin-Ovchinnikov Institute of Bioorganic Chemistry, Miklukho-Maklaya St., 16/10, Moscow, 117997, Russia.
  • Borisevich SS; The Russian Academy of Sciences, Ufa Institute of Chemistry, Octyabrya Av., 71, Ufa, 450078, Russia.
  • Mozhaitsev ES; Siberian Branch of the Russian Academy of Sciences, N. N. Vorozhtsov Novosibirsk Institute of Organic Chemistry, Lavrentiev Av., 9, Novosibirsk, 630090, Russia.
  • Saloutin VI; Ural Branch of the Russian Academy of Sciences, Postovsky Institute of Organic Synthesis, S. Kovalevskoi St., 22, Ekaterinburg, 620108, Russia.
ChemMedChem ; 18(12): e202300063, 2023 06 15.
Article en En | MEDLINE | ID: mdl-37006199

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Canales Catiónicos TRPV / Analgésicos Idioma: En Revista: ChemMedChem Asunto de la revista: FARMACOLOGIA / QUIMICA Año: 2023 Tipo del documento: Article

Texto completo: 1 Base de datos: MEDLINE Asunto principal: Canales Catiónicos TRPV / Analgésicos Idioma: En Revista: ChemMedChem Asunto de la revista: FARMACOLOGIA / QUIMICA Año: 2023 Tipo del documento: Article