1.
Ann N Y Acad Sci
; 971: 139-41, 2002 Oct.
Artículo
en Inglés
| MEDLINE
| ID: mdl-12438104
RESUMEN
Adrenal secretion and binding studies were performed using ring E analogues of methyllycaconitine to assess structural determinants affecting activity on bovine adrenal alpha3beta4* nicotinic receptors. The most potent analogues are as potent as many inhibitors of adrenal secretion. Our data support the potential use of methyllycaconitine analogues to generate nicotinic receptor subtype-specific compounds.