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Bioorg Med Chem Lett
; 17(15): 4284-9, 2007 Aug 01.
Artículo
en Inglés
| MEDLINE
| ID: mdl-17540562
RESUMEN
The identification of a potent series of IKK-beta selective inhibitors based on an imidazothienopyrazine template and the oral efficacy of one such analog (22j) in the LPS-induced TNF-alpha release mouse model are described.