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Histone methyltransferase inhibitors are orally bioavailable, fast-acting molecules with activity against different species causing malaria in humans.
Malmquist, Nicholas A; Sundriyal, Sandeep; Caron, Joachim; Chen, Patty; Witkowski, Benoit; Menard, Didier; Suwanarusk, Rossarin; Renia, Laurent; Nosten, Francois; Jiménez-Díaz, María Belén; Angulo-Barturen, Iñigo; Santos Martínez, María; Ferrer, Santiago; Sanz, Laura M; Gamo, Francisco-Javier; Wittlin, Sergio; Duffy, Sandra; Avery, Vicky M; Ruecker, Andrea; Delves, Michael J; Sinden, Robert E; Fuchter, Matthew J; Scherf, Artur.
Afiliación
  • Malmquist NA; Unité de Biologie des Interactions Hôte-Parasite, Institut Pasteur, Paris, France Centre National de la Recherche Scientifique, Unité de Recherche Associée 2581, Paris, France nicholas.malmquist@pasteur.fr artur.scherf@pasteur.fr.
  • Sundriyal S; Department of Chemistry, Imperial College London, South Kensington Campus, London, United Kingdom.
  • Caron J; Department of Chemistry, Imperial College London, South Kensington Campus, London, United Kingdom.
  • Chen P; Unité de Biologie des Interactions Hôte-Parasite, Institut Pasteur, Paris, France Centre National de la Recherche Scientifique, Unité de Recherche Associée 2581, Paris, France.
  • Witkowski B; Institut Pasteur du Cambodge, Malaria Molecular Epidemiology Unit, Phnom Penh, Cambodia.
  • Menard D; Institut Pasteur du Cambodge, Malaria Molecular Epidemiology Unit, Phnom Penh, Cambodia.
  • Suwanarusk R; Singapore Immunology Network (SIgN), Agency for Science, Technology and Research (A*STAR), Biopolis, Singapore.
  • Renia L; Singapore Immunology Network (SIgN), Agency for Science, Technology and Research (A*STAR), Biopolis, Singapore.
  • Nosten F; Centre for Tropical Medicine, Nuffield Department of Medicine, University of Oxford, Oxford, United Kingdom Shoklo Malaria Research Unit, Mahidol-Oxford Tropical Medicine Research Unit, Faculty of Tropical Medicine, Mahidol University, Mae Sot, Thailand.
  • Jiménez-Díaz MB; Tres Cantos Medicines Development Campus, Diseases of the Developing World, GlaxoSmithKline, Tres Cantos, Madrid, Spain.
  • Angulo-Barturen I; Tres Cantos Medicines Development Campus, Diseases of the Developing World, GlaxoSmithKline, Tres Cantos, Madrid, Spain.
  • Santos Martínez M; Tres Cantos Medicines Development Campus, Diseases of the Developing World, GlaxoSmithKline, Tres Cantos, Madrid, Spain.
  • Ferrer S; Tres Cantos Medicines Development Campus, Diseases of the Developing World, GlaxoSmithKline, Tres Cantos, Madrid, Spain.
  • Sanz LM; Tres Cantos Medicines Development Campus, Diseases of the Developing World, GlaxoSmithKline, Tres Cantos, Madrid, Spain.
  • Gamo FJ; Tres Cantos Medicines Development Campus, Diseases of the Developing World, GlaxoSmithKline, Tres Cantos, Madrid, Spain.
  • Wittlin S; Parasite Chemotherapy Unit, Swiss Tropical and Public Health Institute, Basel, Switzerland University of Basel, Basel, Switzerland.
  • Duffy S; Discovery Biology, Eskitis Institute, Griffith University, Nathan Campus, Brisbane, Queensland, Australia.
  • Avery VM; Discovery Biology, Eskitis Institute, Griffith University, Nathan Campus, Brisbane, Queensland, Australia.
  • Ruecker A; Division of Cell and Molecular Biology, Imperial College London, South Kensington, London, United Kingdom.
  • Delves MJ; Division of Cell and Molecular Biology, Imperial College London, South Kensington, London, United Kingdom.
  • Sinden RE; Division of Cell and Molecular Biology, Imperial College London, South Kensington, London, United Kingdom.
  • Fuchter MJ; Department of Chemistry, Imperial College London, South Kensington Campus, London, United Kingdom.
  • Scherf A; Unité de Biologie des Interactions Hôte-Parasite, Institut Pasteur, Paris, France Centre National de la Recherche Scientifique, Unité de Recherche Associée 2581, Paris, France nicholas.malmquist@pasteur.fr artur.scherf@pasteur.fr.
Antimicrob Agents Chemother ; 59(2): 950-9, 2015 Feb.
Article en En | MEDLINE | ID: mdl-25421480

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Quinazolinas / Azepinas / N-Metiltransferasa de Histona-Lisina / Malaria / Antimaláricos Límite: Animals / Female / Humans Idioma: En Revista: Antimicrob Agents Chemother Año: 2015 Tipo del documento: Article

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Quinazolinas / Azepinas / N-Metiltransferasa de Histona-Lisina / Malaria / Antimaláricos Límite: Animals / Female / Humans Idioma: En Revista: Antimicrob Agents Chemother Año: 2015 Tipo del documento: Article