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Structure-Based Discovery of 1H-Indazole-3-carboxamides as a Novel Structural Class of Human GSK-3 Inhibitors.
Ombrato, Rosella; Cazzolla, Nicola; Mancini, Francesca; Mangano, Giorgina.
Afiliación
  • Ombrato R; R&D, Computational Chemistry Laboratory, ‡Chemistry Department, and §In Vitro Pharmacology Development, Angelini Research Center, ACRAF S.p.A. , Piazzale della Stazione, snc, I-00071 Santa Palomba, Pomezia (RM), Italy.
  • Cazzolla N; R&D, Computational Chemistry Laboratory, ‡Chemistry Department, and §In Vitro Pharmacology Development, Angelini Research Center, ACRAF S.p.A. , Piazzale della Stazione, snc, I-00071 Santa Palomba, Pomezia (RM), Italy.
  • Mancini F; R&D, Computational Chemistry Laboratory, ‡Chemistry Department, and §In Vitro Pharmacology Development, Angelini Research Center, ACRAF S.p.A. , Piazzale della Stazione, snc, I-00071 Santa Palomba, Pomezia (RM), Italy.
  • Mangano G; R&D, Computational Chemistry Laboratory, ‡Chemistry Department, and §In Vitro Pharmacology Development, Angelini Research Center, ACRAF S.p.A. , Piazzale della Stazione, snc, I-00071 Santa Palomba, Pomezia (RM), Italy.
J Chem Inf Model ; 55(12): 2540-51, 2015 Dec 28.
Article en En | MEDLINE | ID: mdl-26600430

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Modelos Moleculares / Dacarbazina / Glucógeno Sintasa Quinasa 3 / Inhibidores Enzimáticos / Descubrimiento de Drogas / Indazoles Límite: Humans Idioma: En Revista: J Chem Inf Model Asunto de la revista: INFORMATICA MEDICA / QUIMICA Año: 2015 Tipo del documento: Article País de afiliación: Italia

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Modelos Moleculares / Dacarbazina / Glucógeno Sintasa Quinasa 3 / Inhibidores Enzimáticos / Descubrimiento de Drogas / Indazoles Límite: Humans Idioma: En Revista: J Chem Inf Model Asunto de la revista: INFORMATICA MEDICA / QUIMICA Año: 2015 Tipo del documento: Article País de afiliación: Italia