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Discovery of Pyrazolopyrimidine Derivatives as Novel Dual Inhibitors of BTK and PI3Kδ.
Pujala, Brahmam; Agarwal, Anil K; Middya, Sandip; Banerjee, Monali; Surya, Arjun; Nayak, Anjan K; Gupta, Ashu; Khare, Sweta; Guguloth, Rambabu; Randive, Nitin A; Shinde, Bharat U; Thakur, Anamika; Patel, Dhananjay I; Raja, Mohd; Green, Michael J; Alfaro, Jennifer; Avila, Patricio; Pérez de Arce, Felipe; Almirez, Ramona G; Kanno, Stacy; Bernales, Sebastián; Hung, David T; Chakravarty, Sarvajit; McCullagh, Emma; Quinn, Kevin P; Rai, Roopa; Pham, Son M.
Afiliación
  • Pujala B; Integral BioSciences, Pvt. Ltd. , C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Agarwal AK; Integral BioSciences, Pvt. Ltd. , C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Middya S; Curadev, Pvt. Ltd. , B-87, Sector 83, Noida, Uttar Pradesh 201305, India.
  • Banerjee M; Curadev, Pvt. Ltd. , B-87, Sector 83, Noida, Uttar Pradesh 201305, India.
  • Surya A; Curadev, Pvt. Ltd. , B-87, Sector 83, Noida, Uttar Pradesh 201305, India.
  • Nayak AK; Integral BioSciences, Pvt. Ltd. , C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Gupta A; Integral BioSciences, Pvt. Ltd. , C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Khare S; Integral BioSciences, Pvt. Ltd. , C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Guguloth R; Integral BioSciences, Pvt. Ltd. , C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Randive NA; Integral BioSciences, Pvt. Ltd. , C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Shinde BU; Integral BioSciences, Pvt. Ltd. , C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Thakur A; Integral BioSciences, Pvt. Ltd. , C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Patel DI; Integral BioSciences, Pvt. Ltd. , C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Raja M; Integral BioSciences, Pvt. Ltd. , C-64, Hosiery Complex Phase II Extension, Noida, Uttar Pradesh 201306, India.
  • Green MJ; Medivation, Inc. , 525 Market Street, 36th Floor, San Francisco, California 94105, United States.
  • Alfaro J; Fundación Ciencia y Vida , Avenida Zañartu 1482, Ñuñoa, Santiago 7780272, Chile.
  • Avila P; Fundación Ciencia y Vida , Avenida Zañartu 1482, Ñuñoa, Santiago 7780272, Chile.
  • Pérez de Arce F; Fundación Ciencia y Vida, Avenida Zañartu 1482, Ñuñoa, Santiago 7780272, Chile; Departamento de Ciencias Biológicas, Facultad de Ciencias Biológicas, Universidad Andrés Bello, Santiago 8370146, Chile.
  • Almirez RG; Medivation, Inc. , 525 Market Street, 36th Floor, San Francisco, California 94105, United States.
  • Kanno S; Medivation, Inc. , 525 Market Street, 36th Floor, San Francisco, California 94105, United States.
  • Bernales S; Medivation, Inc. , 525 Market Street, 36th Floor, San Francisco, California 94105, United States.
  • Hung DT; Medivation, Inc. , 525 Market Street, 36th Floor, San Francisco, California 94105, United States.
  • Chakravarty S; Medivation, Inc. , 525 Market Street, 36th Floor, San Francisco, California 94105, United States.
  • McCullagh E; Medivation, Inc. , 525 Market Street, 36th Floor, San Francisco, California 94105, United States.
  • Quinn KP; Medivation, Inc. , 525 Market Street, 36th Floor, San Francisco, California 94105, United States.
  • Rai R; Medivation, Inc. , 525 Market Street, 36th Floor, San Francisco, California 94105, United States.
  • Pham SM; Medivation, Inc. , 525 Market Street, 36th Floor, San Francisco, California 94105, United States.
ACS Med Chem Lett ; 7(12): 1161-1166, 2016 Dec 08.
Article en En | MEDLINE | ID: mdl-27994757

Texto completo: 1 Banco de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2016 Tipo del documento: Article País de afiliación: India

Texto completo: 1 Banco de datos: MEDLINE Idioma: En Revista: ACS Med Chem Lett Año: 2016 Tipo del documento: Article País de afiliación: India