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Crystallography-guided discovery of carbazole-based retinoic acid-related orphan receptor gamma-t (RORγt) modulators: insights into different protein behaviors with "short" and "long" inverse agonists.
Yu, Ming-Cheng; Yang, Feng; Ding, Xiao-Yu; Sun, Nan-Nan; Jiang, Zheng-Yuan; Huang, Ya-Fei; Yan, Yu-Rong; Zhu, Chen; Xie, Qiong; Chen, Zhi-Feng; Guo, Si-Qi; Jiang, Hua-Liang; Chen, Kai-Xian; Luo, Cheng; Luo, Xiao-Min; Chen, Shi-Jie; Wang, Yong-Hui.
Afiliación
  • Yu MC; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Yang F; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Ding XY; Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China.
  • Sun NN; University of Chinese Academy of Sciences, Beijing, 100049, China.
  • Jiang ZY; Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China.
  • Huang YF; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Yan YR; Key Laboratory of Metabolism and Molecular Medicine, The Ministry of Education, Department of Biochemistry and Molecular Biology, Shanghai Medical College, Fudan University, Shanghai, 200032, China.
  • Zhu C; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Xie Q; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Chen ZF; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Guo SQ; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Jiang HL; Department of Medicinal Chemistry, School of Pharmacy, Fudan University, Shanghai, 201203, China.
  • Chen KX; Fudan Zhangjiang Institute, Shanghai, 201203, China.
  • Luo C; University of Chinese Academy of Sciences, Beijing, 100049, China.
  • Luo XM; Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China.
  • Chen SJ; Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai, 201203, China.
  • Wang YH; University of Chinese Academy of Sciences, Beijing, 100049, China.
Acta Pharmacol Sin ; 42(9): 1524-1534, 2021 Sep.
Article en En | MEDLINE | ID: mdl-33239687
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Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Carbazoles / Receptores de Ácido Retinoico / Cristalografía / Agonismo Inverso de Drogas / Miembro 3 del Grupo F de la Subfamilia 1 de Receptores Nucleares Idioma: En Revista: Acta Pharmacol Sin Asunto de la revista: FARMACOLOGIA Año: 2021 Tipo del documento: Article País de afiliación: China
Texto completo
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Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Carbazoles / Receptores de Ácido Retinoico / Cristalografía / Agonismo Inverso de Drogas / Miembro 3 del Grupo F de la Subfamilia 1 de Receptores Nucleares Idioma: En Revista: Acta Pharmacol Sin Asunto de la revista: FARMACOLOGIA Año: 2021 Tipo del documento: Article País de afiliación: China