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Design, Sustainable Synthesis and Biological Evaluation of a Novel Dual α2A/5-HT7 Receptor Antagonist with Antidepressant-Like Properties.
Canale, Vittorio; Kotanska, Magdalena; Dziubina, Anna; Stefaniak, Matylda; Siwek, Agata; Starowicz, Gabriela; Marciniec, Krzysztof; Kasza, Patryk; Satala, Grzegorz; Duszynska, Beata; Bantreil, Xavier; Lamaty, Frédéric; Bednarski, Marek; Sapa, Jacek; Zajdel, Pawel.
Afiliación
  • Canale V; Department of Organic Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, 30-688 Kraków, Poland.
  • Kotanska M; Department of Pharmacodynamics, Faculty of Pharmacy, Jagiellonian University Medical College, 30-688 Kraków, Poland.
  • Dziubina A; Department of Pharmacodynamics, Faculty of Pharmacy, Jagiellonian University Medical College, 30-688 Kraków, Poland.
  • Stefaniak M; Department of Organic Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, 30-688 Kraków, Poland.
  • Siwek A; Department of Pharmacobiology, Faculty of Pharmacy, Jagiellonian University Medical College, 30-688 Kraków, Poland.
  • Starowicz G; Department of Pharmacobiology, Faculty of Pharmacy, Jagiellonian University Medical College, 30-688 Kraków, Poland.
  • Marciniec K; Department of Organic Chemistry, Medical University of Silesia, 41-200 Sosnowiec, Poland.
  • Kasza P; Department of Organic Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, 30-688 Kraków, Poland.
  • Satala G; Department of Medicinal Chemistry, Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343 Kraków, Poland.
  • Duszynska B; Department of Medicinal Chemistry, Maj Institute of Pharmacology, Polish Academy of Sciences, 31-343 Kraków, Poland.
  • Bantreil X; IBMM, Université de Montpellier, CNRS, ENSCM, 34095 Montpellier, France.
  • Lamaty F; IBMM, Université de Montpellier, CNRS, ENSCM, 34095 Montpellier, France.
  • Bednarski M; Department of Pharmacodynamics, Faculty of Pharmacy, Jagiellonian University Medical College, 30-688 Kraków, Poland.
  • Sapa J; Department of Pharmacodynamics, Faculty of Pharmacy, Jagiellonian University Medical College, 30-688 Kraków, Poland.
  • Zajdel P; Department of Organic Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, 30-688 Kraków, Poland.
Molecules ; 26(13)2021 Jun 23.
Article en En | MEDLINE | ID: mdl-34201675

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Receptores de Serotonina / Receptores Adrenérgicos alfa 2 / Depresión / Antagonistas de Receptores Adrenérgicos alfa 2 / Actividad Motora / Antidepresivos Tipo de estudio: Prognostic_studies Límite: Animals / Humans / Male Idioma: En Revista: Molecules Asunto de la revista: BIOLOGIA Año: 2021 Tipo del documento: Article País de afiliación: Polonia

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Receptores de Serotonina / Receptores Adrenérgicos alfa 2 / Depresión / Antagonistas de Receptores Adrenérgicos alfa 2 / Actividad Motora / Antidepresivos Tipo de estudio: Prognostic_studies Límite: Animals / Humans / Male Idioma: En Revista: Molecules Asunto de la revista: BIOLOGIA Año: 2021 Tipo del documento: Article País de afiliación: Polonia