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Discovery of new pyridine-quinoline hybrids as competitive and non-competitive PIM-1 kinase inhibitors with apoptosis induction and caspase 3/7 activation capabilities.
El-Miligy, Mostafa M M; Abdelaziz, Marwa E; Fahmy, Salwa M; Ibrahim, Tamer M; Abu-Serie, Marwa M; Mahran, Mona A; Hazzaa, Aly A.
Afiliación
  • El-Miligy MMM; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Alexandria University, Alexandria, Egypt.
  • Abdelaziz ME; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Alexandria University, Alexandria, Egypt.
  • Fahmy SM; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Alexandria University, Alexandria, Egypt.
  • Ibrahim TM; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Kafrelsheikh University, Kafrelsheikh, Egypt.
  • Abu-Serie MM; Medical Biotechnology Department, Genetic Engineering and Biotechnology Research Institute (GEBRI, City of Scientific Research and Technological Applications (SRTA-City), Alexandria, Egypt).
  • Mahran MA; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Alexandria University, Alexandria, Egypt.
  • Hazzaa AA; Pharmaceutical Chemistry Department, Faculty of Pharmacy, Alexandria University, Alexandria, Egypt.
J Enzyme Inhib Med Chem ; 38(1): 2152810, 2023 Dec.
Article en En | MEDLINE | ID: mdl-36629075

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Quinolinas / Antineoplásicos Límite: Humans / Male Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Egipto

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Quinolinas / Antineoplásicos Límite: Humans / Male Idioma: En Revista: J Enzyme Inhib Med Chem Asunto de la revista: BIOQUIMICA / QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Egipto