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Design and Synthesis of Novel Cereblon Binders for Use in Targeted Protein Degradation.
Norris, Stephen; Ba, Xiaochu; Rhodes, Jayce; Huang, Dehua; Khambatta, Gody; Buenviaje, Jennifer; Nayak, Surendra; Meiring, Joseph; Reiss, Samantha; Xu, Shuichan; Shi, Lihong; Whitefield, Brandon; Alexander, Matt; Horn, Evan J; Correa, Matthew; Tehrani, Lida; Hansen, Joshua D; Papa, Patrick; Mortensen, Deborah S.
Afiliación
  • Norris S; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Ba X; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Rhodes J; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Huang D; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Khambatta G; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Buenviaje J; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Nayak S; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Meiring J; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Reiss S; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Xu S; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Shi L; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Whitefield B; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Alexander M; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Horn EJ; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Correa M; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Tehrani L; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Hansen JD; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Papa P; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Mortensen DS; Bristol Myers Squibb, 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
J Med Chem ; 66(23): 16388-16409, 2023 12 14.
Article en En | MEDLINE | ID: mdl-37991844

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Péptido Hidrolasas / Ubiquitina-Proteína Ligasas Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Banco de datos: MEDLINE Asunto principal: Péptido Hidrolasas / Ubiquitina-Proteína Ligasas Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2023 Tipo del documento: Article País de afiliación: Estados Unidos