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1.
Genetic complexity alters drug susceptibility of asexual and gametocyte stages of Plasmodium falciparum to antimalarial candidates.
Antimicrob Agents Chemother
; 68(3): e0129123, 2024 Mar 06.
Article
in English
| MEDLINE | ID: mdl-38259087
2.
A Dynamic and Combinatorial Histone Code Drives Malaria Parasite Asexual and Sexual Development.
Mol Cell Proteomics
; 21(3): 100199, 2022 03.
Article
in English
| MEDLINE | ID: mdl-35051657
3.
New Transmission-Selective Antimalarial Agents through Hit-to-Lead Optimization of 2-([1,1'-Biphenyl]-4-carboxamido)benzoic Acid Derivatives.
Chembiochem
; 23(21): e202200427, 2022 11 04.
Article
in English
| MEDLINE | ID: mdl-36106425
4.
The ecdysone receptor regulates several key physiological factors in Anopheles funestus.
Malar J
; 21(1): 97, 2022 Mar 19.
Article
in English
| MEDLINE | ID: mdl-35305668
5.
MALBoost: a web-based application for gene regulatory network analysis in Plasmodium falciparum.
Malar J
; 20(1): 317, 2021 Jul 14.
Article
in English
| MEDLINE | ID: mdl-34261498
6.
Parasite genetic diversity reflects continued residual malaria transmission in Vhembe District, a hotspot in the Limpopo Province of South Africa.
Malar J
; 20(1): 96, 2021 Feb 16.
Article
in English
| MEDLINE | ID: mdl-33593382
7.
Poly(N-vinylpyrrolidone) Antimalaria Conjugates of Membrane-Disruptive Peptides.
Biomacromolecules
; 21(12): 5053-5066, 2020 12 14.
Article
in English
| MEDLINE | ID: mdl-33156615
8.
High levels of imported asymptomatic malaria but limited local transmission in KwaZulu-Natal, a South African malaria-endemic province nearing malaria elimination.
Malar J
; 19(1): 152, 2020 Apr 15.
Article
in English
| MEDLINE | ID: mdl-32295590
9.
Hierarchical transcriptional control regulates Plasmodium falciparum sexual differentiation.
BMC Genomics
; 20(1): 920, 2019 Dec 03.
Article
in English
| MEDLINE | ID: mdl-31795940
10.
Bioassay-guided isolation and identification of gametocytocidal compounds from Artemisia afra (Asteraceae).
Malar J
; 18(1): 65, 2019 Mar 08.
Article
in English
| MEDLINE | ID: mdl-30849984
11.
Artemisone and Artemiside Are Potent Panreactive Antimalarial Agents That Also Synergize Redox Imbalance in Plasmodium falciparum Transmissible Gametocyte Stages.
Antimicrob Agents Chemother
; 62(8)2018 08.
Article
in English
| MEDLINE | ID: mdl-29866868
12.
UCT943, a Next-Generation Plasmodium falciparum PI4K Inhibitor Preclinical Candidate for the Treatment of Malaria.
Antimicrob Agents Chemother
; 62(9)2018 09.
Article
in English
| MEDLINE | ID: mdl-29941635
13.
Potent Plasmodium falciparum gametocytocidal compounds identified by exploring the kinase inhibitor chemical space for dual active antimalarials.
J Antimicrob Chemother
; 73(5): 1279-1290, 2018 05 01.
Article
in English
| MEDLINE | ID: mdl-29420756
14.
Understanding human genetic factors influencing primaquine safety and efficacy to guide primaquine roll-out in a pre-elimination setting in southern Africa.
Malar J
; 17(1): 120, 2018 Mar 20.
Article
in English
| MEDLINE | ID: mdl-29558929
15.
Synthesis, antimalarial activities and cytotoxicities of amino-artemisinin-1,2-disubstituted ferrocene hybrids.
Bioorg Med Chem Lett
; 28(19): 3161-3163, 2018 10 15.
Article
in English
| MEDLINE | ID: mdl-30174153
16.
Synthesis, in vitro antimalarial activities and cytotoxicities of amino-artemisinin-ferrocene derivatives.
Bioorg Med Chem Lett
; 28(3): 289-292, 2018 02 01.
Article
in English
| MEDLINE | ID: mdl-29317166
17.
Straightforward conversion of decoquinate into inexpensive tractable new derivatives with significant antimalarial activities.
Bioorg Med Chem Lett
; 26(13): 3006-3009, 2016 07 01.
Article
in English
| MEDLINE | ID: mdl-27210430
18.
A novel inhibitor of Plasmodium falciparum spermidine synthase: a twist in the tail.
Malar J
; 14: 54, 2015 Feb 05.
Article
in English
| MEDLINE | ID: mdl-25651815
19.
Nowhere to hide: interrogating different metabolic parameters of Plasmodium falciparum gametocytes in a transmission blocking drug discovery pipeline towards malaria elimination.
Malar J
; 14: 213, 2015 May 22.
Article
in English
| MEDLINE | ID: mdl-25994518
20.
Interrogating alkyl and arylalkylpolyamino (bis)urea and (bis)thiourea isosteres as potent antimalarial chemotypes against multiple lifecycle forms of Plasmodium falciparum parasites.
Bioorg Med Chem
; 23(16): 5131-43, 2015 Aug 15.
Article
in English
| MEDLINE | ID: mdl-25684422