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1.
Comparative Study of Batch and Continuous Flow Reactors in Selective Hydrogenation of Functional Groups in Organic Compounds: What Is More Effective?
Int J Mol Sci
; 24(18)2023 Sep 15.
Article
in English
| MEDLINE | ID: mdl-37762440
2.
Effect of Phosphorus Precursor, Reduction Temperature, and Support on the Catalytic Properties of Nickel Phosphide Catalysts in Continuous-Flow Reductive Amination of Ethyl Levulinate.
Int J Mol Sci
; 23(3)2022 Jan 20.
Article
in English
| MEDLINE | ID: mdl-35163029
3.
Identification of potent inhibitors of the sortilin-progranulin interaction.
Bioorg Med Chem Lett
; 30(17): 127403, 2020 09 01.
Article
in English
| MEDLINE | ID: mdl-32738972
4.
Structural characterization of nonactive site, TrkA-selective kinase inhibitors.
Proc Natl Acad Sci U S A
; 114(3): E297-E306, 2017 01 17.
Article
in English
| MEDLINE | ID: mdl-28039433
5.
Two-Step One-Pot Reductive Amination of Furanic Aldehydes Using CuAlOx Catalyst in a Flow Reactor.
Molecules
; 25(20)2020 Oct 17.
Article
in English
| MEDLINE | ID: mdl-33080807
6.
Cerastecins inhibit membrane lipooligosaccharide transport in drug-resistant Acinetobacter baumannii.
Nat Microbiol
; 9(5): 1244-1255, 2024 May.
Article
in English
| MEDLINE | ID: mdl-38649414
7.
Potent targeted activator of cell kill molecules eliminate cells expressing HIV-1.
Sci Transl Med
; 15(684): eabn2038, 2023 02 22.
Article
in English
| MEDLINE | ID: mdl-36812345
8.
Discovery of a novel class of non-ATP site DFG-out state p38 inhibitors utilizing computationally assisted virtual fragment-based drug design (vFBDD).
Bioorg Med Chem Lett
; 21(23): 7155-65, 2011 Dec 01.
Article
in English
| MEDLINE | ID: mdl-22014550
9.
Discovery of an Anion-Dependent Farnesyltransferase Inhibitor from a Phenotypic Screen.
ACS Med Chem Lett
; 12(1): 99-106, 2021 Jan 14.
Article
in English
| MEDLINE | ID: mdl-33488970
10.
Analysis of imatinib and sorafenib binding to p38alpha compared with c-Abl and b-Raf provides structural insights for understanding the selectivity of inhibitors targeting the DFG-out form of protein kinases.
Biochemistry
; 49(17): 3611-8, 2010 May 04.
Article
in English
| MEDLINE | ID: mdl-20337484
11.
The rational design of a novel potent analogue of the 5'-AMP-activated protein kinase inhibitor compound C with improved selectivity and cellular activity.
Bioorg Med Chem Lett
; 20(22): 6394-9, 2010 Nov 15.
Article
in English
| MEDLINE | ID: mdl-20932747
12.
Discovery and SAR of a series of 4,6-diamino-1,3,5-triazin-2-ol as novel non-nucleoside reverse transcriptase inhibitors of HIV-1.
Bioorg Med Chem Lett
; 20(22): 6592-6, 2010 Nov 15.
Article
in English
| MEDLINE | ID: mdl-20888224
13.
Structure-based design of substituted biphenyl ethylene ethers as ligands binding in the hydrophobic pocket of gp41 and blocking the helical bundle formation.
Bioorg Med Chem Lett
; 19(19): 5693-7, 2009 Oct 01.
Article
in English
| MEDLINE | ID: mdl-19699090
14.
Hepatitis C virus NS3 protease requires its NS4A cofactor peptide for optimal binding of a boronic acid inhibitor as shown by NMR.
Chem Biol
; 9(1): 79-92, 2002 Jan.
Article
in English
| MEDLINE | ID: mdl-11841941
15.
Synthesis and pharmacological evaluation of N-(3-(1H-indol-4-yl)-5-(2-methoxyisonicotinoyl)phenyl)methanesulfonamide (LP-261), a potent antimitotic agent.
J Med Chem
; 54(1): 179-200, 2011 Jan 13.
Article
in English
| MEDLINE | ID: mdl-21126027
16.
Mutagenesis of p38alpha MAP kinase establishes key roles of Phe169 in function and structural dynamics and reveals a novel DFG-OUT state.
Biochemistry
; 46(19): 5687-96, 2007 May 15.
Article
in English
| MEDLINE | ID: mdl-17441692
17.
Two classes of p38alpha MAP kinase inhibitors having a common diphenylether core but exhibiting divergent binding modes.
Bioorg Med Chem Lett
; 15(23): 5274-9, 2005 Dec 01.
Article
in English
| MEDLINE | ID: mdl-16169718
18.
A Biacore biosensor method for detailed kinetic binding analysis of small molecule inhibitors of p38alpha mitogen-activated protein kinase.
Anal Biochem
; 325(1): 126-36, 2004 Feb 01.
Article
in English
| MEDLINE | ID: mdl-14715293
19.
Improved expression, purification, and crystallization of p38alpha MAP kinase.
Protein Expr Purif
; 37(1): 154-61, 2004 Sep.
Article
in English
| MEDLINE | ID: mdl-15294293
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