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1.
Novel and Potent Small Molecules against Melanoma Harboring BRAF Class I/II/III Mutants for Overcoming Drug Resistance.
Int J Mol Sci
; 22(7)2021 Apr 06.
Article
in English
| MEDLINE | ID: mdl-33917428
2.
Affinity-Directed Site-Specific Protein Labeling and Its Application to Antibody-Drug Conjugates.
Adv Sci (Weinh)
; 11(4): e2306401, 2024 Jan.
Article
in English
| MEDLINE | ID: mdl-38032124
3.
Correction: Nam et al. Identification of Thiazolo[5,4-b]pyridine Derivatives as c-KIT Inhibitors for Overcoming Imatinib Resistance. Cancers 2023, 15, 143.
Cancers (Basel)
; 16(11)2024 Jun 06.
Article
in English
| MEDLINE | ID: mdl-38893284
4.
Synthesis and antibacterial activities of baulamycin A inspired derivatives.
Eur J Med Chem
; 259: 115592, 2023 Nov 05.
Article
in English
| MEDLINE | ID: mdl-37478559
5.
Identification of Pyrido[3,4-d]pyrimidine derivatives as RIPK3-Mediated necroptosis inhibitors.
Eur J Med Chem
; 259: 115635, 2023 Nov 05.
Article
in English
| MEDLINE | ID: mdl-37494773
6.
Targeted kinase degradation via the KLHDC2 ubiquitin E3 ligase.
Cell Chem Biol
; 30(11): 1414-1420.e5, 2023 11 16.
Article
in English
| MEDLINE | ID: mdl-37567174
7.
Identification of Pyridinyltriazine Derivatives as Potent panFGFR Inhibitors against Gatekeeper Mutants for Overcoming Drug Resistance.
J Med Chem
; 65(8): 6017-6038, 2022 04 28.
Article
in English
| MEDLINE | ID: mdl-35436119
8.
Identification of Thiazolo[5,4-b]pyridine Derivatives as c-KIT Inhibitors for Overcoming Imatinib Resistance.
Cancers (Basel)
; 15(1)2022 Dec 26.
Article
in English
| MEDLINE | ID: mdl-36612139
9.
Novel Macrocyclic Peptidomimetics Targeting the Polo-Box Domain of Polo-Like Kinase 1.
J Med Chem
; 65(3): 1915-1932, 2022 02 10.
Article
in English
| MEDLINE | ID: mdl-35029981
10.
Anti-Tumor Activity of AZD4547 Against NTRK1 Fusion Positive Cancer Cells Through Inhibition of NTRKs.
Front Oncol
; 11: 757598, 2021.
Article
in English
| MEDLINE | ID: mdl-34790577
11.
Novel Small Molecules Capable of Blocking mtRAS-Signaling Pathway.
Front Oncol
; 11: 768022, 2021.
Article
in English
| MEDLINE | ID: mdl-34956887
12.
Procaspase activating compound 1 controls tetracycline repressor-regulated gene expression system.
Biosci Rep
; 39(1)2019 01 31.
Article
in English
| MEDLINE | ID: mdl-30538170
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