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Bioorg Med Chem Lett
; 27(9): 2023-2028, 2017 05 01.
Artículo
en Inglés
| MEDLINE
| ID: mdl-28336141
RESUMEN
A series of potent, competitive and highly selective kynurenine monooxygenase inhibitors have been discovered via a substrate-based approach for the treatment of acute pancreatitis. The lead compound demonstrated good cellular potency and clear pharmacodynamic activity in vivo.