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Design, synthesis and evaluation of antiestrogen and histone deacetylase inhibitor molecular hybrids.
Mendoza-Sanchez, Rodrigo; Cotnoir-White, David; Kulpa, Justyna; Jutras, Isabel; Pottel, Joshua; Moitessier, Nicolas; Mader, Sylvie; Gleason, James L.
Affiliation
  • Mendoza-Sanchez R; Department of Chemistry, Otto Maass Building, McGill University, 801 Sherbrooke Street West, Montreal, Québec H3A 0B8, Canada.
  • Cotnoir-White D; Institute for Research in Immunology and Cancer, Pavillon Marcelle-Coutu, Université de Montréal, 2950 chemin de Polytechnique, Montréal, Québec H3T 1J4, Canada.
  • Kulpa J; Institute for Research in Immunology and Cancer, Pavillon Marcelle-Coutu, Université de Montréal, 2950 chemin de Polytechnique, Montréal, Québec H3T 1J4, Canada.
  • Jutras I; Institute for Research in Immunology and Cancer, Pavillon Marcelle-Coutu, Université de Montréal, 2950 chemin de Polytechnique, Montréal, Québec H3T 1J4, Canada.
  • Pottel J; Department of Chemistry, Otto Maass Building, McGill University, 801 Sherbrooke Street West, Montreal, Québec H3A 0B8, Canada.
  • Moitessier N; Department of Chemistry, Otto Maass Building, McGill University, 801 Sherbrooke Street West, Montreal, Québec H3A 0B8, Canada.
  • Mader S; Institute for Research in Immunology and Cancer, Pavillon Marcelle-Coutu, Université de Montréal, 2950 chemin de Polytechnique, Montréal, Québec H3T 1J4, Canada. Electronic address: sylvie.mader@umontreal.ca.
  • Gleason JL; Department of Chemistry, Otto Maass Building, McGill University, 801 Sherbrooke Street West, Montreal, Québec H3A 0B8, Canada. Electronic address: jim.gleason@mcgill.ca.
Bioorg Med Chem ; 23(24): 7597-606, 2015 Dec 15.
Article in En | MEDLINE | ID: mdl-26613635

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Breast Neoplasms / Estrogen Receptor Modulators / Histone Deacetylase Inhibitors / Antineoplastic Agents Limits: Female / Humans Language: En Journal: Bioorg Med Chem Journal subject: BIOQUIMICA / QUIMICA Year: 2015 Type: Article Affiliation country: Canada

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Breast Neoplasms / Estrogen Receptor Modulators / Histone Deacetylase Inhibitors / Antineoplastic Agents Limits: Female / Humans Language: En Journal: Bioorg Med Chem Journal subject: BIOQUIMICA / QUIMICA Year: 2015 Type: Article Affiliation country: Canada