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Structural Characterization of the Interaction of the Fibroblast Growth Factor Receptor with a Small Molecule Allosteric Inhibitor.
Kappert, Franziska; Sreeramulu, Sridhar; Jonker, Hendrik R A; Richter, Christian; Rogov, Vladimir V; Proschak, Ewgenij; Hargittay, Bruno; Saxena, Krishna; Schwalbe, Harald.
Affiliation
  • Kappert F; Goethe University, Center for Biomolecular Magnetic Resonance (BMRZ), Institute for Organic Chemistry and Chemical Biology, Max von Laue-Straße 7, 60438, Frankfurt am Main, Germany.
  • Sreeramulu S; Goethe University, Center for Biomolecular Magnetic Resonance (BMRZ), Institute for Organic Chemistry and Chemical Biology, Max von Laue-Straße 7, 60438, Frankfurt am Main, Germany.
  • Jonker HRA; Goethe University, Center for Biomolecular Magnetic Resonance (BMRZ), Institute for Organic Chemistry and Chemical Biology, Max von Laue-Straße 7, 60438, Frankfurt am Main, Germany.
  • Richter C; Goethe University, Center for Biomolecular Magnetic Resonance (BMRZ), Institute for Organic Chemistry and Chemical Biology, Max von Laue-Straße 7, 60438, Frankfurt am Main, Germany.
  • Rogov VV; Goethe University, Center for Biomolecular Magnetic Resonance (BMRZ), Institute for Biophysical Chemistry, Max von Laue-Straße 9, 60438, Frankfurt am Main, Germany.
  • Proschak E; Goethe University, Institute of Pharmaceutical Chemistry, Max von Laue-Straße 9, 60438, Frankfurt, Germany.
  • Hargittay B; Goethe University, Center for Biomolecular Magnetic Resonance (BMRZ), Institute for Organic Chemistry and Chemical Biology, Max von Laue-Straße 7, 60438, Frankfurt am Main, Germany.
  • Saxena K; Goethe University, Center for Biomolecular Magnetic Resonance (BMRZ), Institute for Organic Chemistry and Chemical Biology, Max von Laue-Straße 7, 60438, Frankfurt am Main, Germany.
  • Schwalbe H; German Cancer Research Center (DKFZ), Partner facility Frankfurt/Mainz.
Chemistry ; 24(31): 7861-7865, 2018 Jun 04.
Article in En | MEDLINE | ID: mdl-29656465

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Receptors, Fibroblast Growth Factor / Protein Kinase Inhibitors / Ortho-Aminobenzoates / Indolizines / Antineoplastic Agents Type of study: Prognostic_studies Language: En Journal: Chemistry Journal subject: QUIMICA Year: 2018 Type: Article Affiliation country: Germany

Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Receptors, Fibroblast Growth Factor / Protein Kinase Inhibitors / Ortho-Aminobenzoates / Indolizines / Antineoplastic Agents Type of study: Prognostic_studies Language: En Journal: Chemistry Journal subject: QUIMICA Year: 2018 Type: Article Affiliation country: Germany