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Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain (BET) Inhibitors Targeting a Methionine.
Kharenko, Olesya A; Patel, Reena G; Brown, S David; Calosing, Cyrus; White, Andre; Lakshminarasimhan, Damodharan; Suto, Robert K; Duffy, Bryan C; Kitchen, Douglas B; McLure, Kevin G; Hansen, Henrik C; van der Horst, Edward H; Young, Peter R.
Affiliation
  • Kharenko OA; Zenith Epigenetics , Suite 300, 4820 Richard Road SW , Calgary , Alberta T3E 6L1 , Canada.
  • Patel RG; Zenith Epigenetics , Suite 300, 4820 Richard Road SW , Calgary , Alberta T3E 6L1 , Canada.
  • Brown SD; Zenith Epigenetics , Suite 300, 4820 Richard Road SW , Calgary , Alberta T3E 6L1 , Canada.
  • Calosing C; Zenith Epigenetics , Suite 300, 4820 Richard Road SW , Calgary , Alberta T3E 6L1 , Canada.
  • White A; Xtal BioStructures, Inc. , 12 Michigan Drive , Natick , Massachusetts 01760 , United States.
  • Lakshminarasimhan D; Xtal BioStructures, Inc. , 12 Michigan Drive , Natick , Massachusetts 01760 , United States.
  • Suto RK; Xtal BioStructures, Inc. , 12 Michigan Drive , Natick , Massachusetts 01760 , United States.
  • Duffy BC; AMRI , 26 Corporate Circle , P.O. Box 15098, Albany , New York 12212-5098 , United States.
  • Kitchen DB; AMRI , 26 Corporate Circle , P.O. Box 15098, Albany , New York 12212-5098 , United States.
  • McLure KG; Zenith Epigenetics , Suite 300, 4820 Richard Road SW , Calgary , Alberta T3E 6L1 , Canada.
  • Hansen HC; Zenith Epigenetics , Suite 300, 4820 Richard Road SW , Calgary , Alberta T3E 6L1 , Canada.
  • van der Horst EH; Zenith Epigenetics , Suite 300, 4820 Richard Road SW , Calgary , Alberta T3E 6L1 , Canada.
  • Young PR; Zenith Epigenetics , Suite 300, 4820 Richard Road SW , Calgary , Alberta T3E 6L1 , Canada.
J Med Chem ; 61(18): 8202-8211, 2018 09 27.
Article in En | MEDLINE | ID: mdl-30165024
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Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Transcription Factors / Nuclear Proteins / Drug Design / Hematologic Neoplasms / Drug Discovery / Methionine / Antineoplastic Agents Type of study: Prognostic_studies Limits: Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2018 Type: Article Affiliation country: Canada
Fulltext
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PubMed Links
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Full text: 1 Collection: 01-internacional Database: MEDLINE Main subject: Transcription Factors / Nuclear Proteins / Drug Design / Hematologic Neoplasms / Drug Discovery / Methionine / Antineoplastic Agents Type of study: Prognostic_studies Limits: Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2018 Type: Article Affiliation country: Canada